| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTK2 |
2-(2-Pyridyl)benzimidazole |
NA |
NA |
NA |
103000 |
NA |
NA |
BindingDB |
| PTK2 |
N-[2-[[4-(trifluoromethyl)-6-(3,4,5-trimethoxyanilino)-1,3,5-triazin-2-yl]amino]phenyl]acetamide |
NA |
125600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTK2 |
4-(1,3-Oxazol-5-yl)pyridine |
NA |
NA |
1350000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTK2 |
2-Acetamido-5-chloropyridine |
NA |
NA |
719000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTK2 |
3-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-2-carboxylic acid |
NA |
NA |
460000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTK6 |
3-[(6-bromo-9H-pyrido[2,3-b]indol-4-yl)amino]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
3-[[6-[4-(2-hydroxyethyl)piperazin-1-yl]sulfonyl-9H-pyrido[2,3-b]indol-4-yl]amino]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
N-(2-methylphenyl)-9H-pyrido[2,3-b]indol-4-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
3-[(6-morpholin-4-ylsulfonyl-9H-pyrido[2,3-b]indol-4-yl)amino]phenol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
1-[4-(3-hydroxyanilino)-9H-pyrido[2,3-b]indol-6-yl]ethanone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
N-(4-chlorophenyl)-9H-pyrido[2,3-b]indol-4-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTK6 |
2-cyano-N-(2,5-dibromophenyl)-3-oxobutanamide |
NA |
267000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTP4A1 |
Rhodanine |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTP4A1 |
CK2/Pim1-IN-1 |
NA |
209000 |
NA |
NA |
NA |
NA |
TTD |
| PTP4A1 |
8-Carboxy-2-phenyl[1,3]thiazolo[3,2-a]pyridin-4-ium-3-olate |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTP4A1 |
propan-2-yl (Z)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate |
NA |
133200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTP4A2 |
Rhodanine |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTP4A2 |
CK2/Pim1-IN-1 |
NA |
188000 |
NA |
NA |
NA |
NA |
TTD |
| PTP4A2 |
8-Carboxy-2-phenyl[1,3]thiazolo[3,2-a]pyridin-4-ium-3-olate |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTP4A2 |
propan-2-yl (Z)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate |
NA |
149800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |