Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN1 4-[4-(2-Benzyl-1-benzofuran-3-yl)phenyl]-2-bromophenol NA 275000000|275422870.3 NA NA NA NA BindingDB|TTD
PTPN1 2-[4-[4-(2-Benzyl-1-benzothiophen-3-yl)phenyl]-2-phenylphenoxy]acetic acid NA 48900000|99900000 NA NA NA NA BindingDB
PTPN1 (2S)-2-[4-[4-[2-[(4-fluorophenyl)methyl]-1-benzofuran-3-yl]phenyl]phenoxy]-3-phenylpropanoic acid NA 602000000|602559586.1 NA NA NA NA BindingDB|TTD
PTPN1 2-[4-[4-(1-Benzofuran-3-yl)phenyl]phenoxy]-3-phenylpropanoic acid NA 288000000|288403150.3 NA NA NA NA BindingDB|TTD
PTPN1 4-((3-(4''-Hydroxybiphenyl-4-yl)benzo[b]thiophen-2-yl)methyl)benzene-1,3-diol NA 588000000 NA NA NA NA BindingDB
PTPN1 2-(4''-(2-Benzylbenzofuran-3-yl)-4-phenethoxybiphenyl-3-ylamino)acetic acid NA 83100000 NA NA NA NA BindingDB
PTPN1 4-[4-(1-Benzofuran-3-yl)phenyl]phenol NA 19900000|19952623.15 NA NA NA NA BindingDB|TTD
PTPN1 2-Butyl-3-[4-(4-methoxyphenyl)phenyl]-1-benzofuran NA 165000000|165958690.7 NA NA NA NA BindingDB|TTD
PTPN1 2-[4'-(2-Butyl-benzofuran-3-yl)-biphenyl-4-yloxy]-3-phenyl-propionic acid NA 436000000 NA NA NA NA BindingDB
PTPN1 (2R)-2-[4-[4-(2-benzyl-1-benzofuran-3-yl)phenyl]phenoxy]-2-phenylacetic acid NA 407000000 NA NA NA NA BindingDB
PTPN1 2-[4'-(2-Bromo-benzofuran-3-yl)-biphenyl-4-yloxy]-3-phenyl-propionic acid NA 407000000|407380277.8 NA NA NA NA BindingDB|TTD
PTPN1 (2S)-2-[4-[4-(2-benzyl-1-benzofuran-3-yl)phenyl]-2-propylphenoxy]-3-phenylpropanoic acid NA 831000000|831763771.1 NA NA NA NA BindingDB|TTD
PTPN1 (2R)-2-[4-[4-[2-[(3,4-dimethoxyphenyl)methyl]-1-benzothiophen-3-yl]phenyl]phenoxy]-3-phenylpropanoic acid NA 120000000 NA NA NA NA BindingDB
PTPN1 (2R)-2-[4-[4-(1-benzylbenzimidazol-2-yl)phenyl]phenoxy]-3-phenylpropanoic acid NA 436000000|436515832.2 NA NA NA NA BindingDB|TTD
PTPN1 Difluoro(naphthalen-2-yl)methanesulfonate NA 175000 NA NA NA NA BindingDB|TTD
PTPN1 Phthalonic acid NA 1500000 NA NA NA NA BindingDB|TTD
PTPN1 (2S)-2-[4'-(2-benzyl-benzofuran-3-yl)-biphenyl-4-yloxy]-3-phenyl-propionic acid methyl ester NA 588000000|588843655.4 NA NA NA NA BindingDB|TTD
PTPN1 4-[4-(2-Ethyl-1-benzofuran-3-yl)phenyl]phenol NA 31600000|31622776.6 NA NA NA NA BindingDB|TTD
PTPN1 Coumarin-3-Carboxylic Acid NA 1000000 NA NA NA NA TTD
PTPN1 2-Chloroacetophenone 480000 NA NA NA NA NA BindingDB|PubChem|TTD