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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTP4A2 ethyl (2E)-2-cyano-3-(3,5-dibromo-4-hydroxyphenyl)prop-2-enoate NA 109200 NA NA NA NA BindingDB|TTD
PTP4A2 prop-2-enyl (E)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate NA 104000 NA NA NA NA BindingDB|TTD
PTP4A2 Thienopyridone NA 104000 NA NA NA NA BindingDB
PTP4A3 8-Carboxy-2-phenyl[1,3]thiazolo[3,2-a]pyridin-4-ium-3-olate NA 102000 NA NA NA NA BindingDB|TTD
PTP4A3 propan-2-yl (Z)-3-(3-bromo-4-hydroxyphenyl)-2-cyanoprop-2-enoate NA 167100 NA NA NA NA BindingDB|TTD
PTP4A3 ethyl (2E)-2-cyano-3-(3,5-dibromo-4-hydroxyphenyl)prop-2-enoate NA 109200 NA NA NA NA BindingDB|TTD
PTPN1 Difluoro-(3-phenylphenyl)methanesulfonic acid NA 115000 NA NA NA NA BindingDB|TTD
PTPN1 2-{3,5-Dibromo-4''''-[5-methyl-2-(4-trifluoromethyl-phenyl)-oxazol-4-yl]-biphenyl-4-yloxy}-3-phenyl-propionic acid NA 131000000|131825673.9 NA NA NA NA BindingDB|TTD
PTPN1 1-Iodyl-4-nitro-benzene NA 130000 NA NA NA NA BindingDB|TTD
PTPN1 Iodoxybenzene NA 2650000 NA NA NA NA BindingDB|TTD
PTPN1 2-(Carboxyformamido)-3-methylbenzoic acid 1090000|1100000|1258925.41 NA NA NA NA NA BindingDB|TTD
PTPN1 Difluoro(1-naphthyl)methylphosphonic acid NA 112000 NA NA NA NA TTD
PTPN1 1-Iodyl-3-nitro-benzene NA 1140000 NA NA NA NA BindingDB|TTD
PTPN1 4-[3-[5-Methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]phenyl]phenol NA 9990000|10000000 NA NA NA NA BindingDB|TTD
PTPN1 Phosphonic acid, (difluoro-2-naphthalenylmethyl)- NA|179000|197000 718100|NA NA NA NA NA BindingDB
PTPN1 2-[4-[3-[5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl]phenyl]phenoxy]acetic Acid NA 63000000|63095734.45 NA NA NA NA BindingDB|TTD
PTPN1 Oleanolic Acid NA 2390000 NA NA NA NA BindingDB|PubChem
PTPN1 4'-(2-Benzyl-benzofuran-3-yl)-3,5-dibromo-biphenyl-4-ol NA 478000000|478630092.3 NA NA NA NA BindingDB|TTD
PTPN1 4'-(2-Benzyl-benzo[b]thiophen-3-yl)-biphenyl-4-ol NA 93300000|275000000|93325430.08 NA NA NA NA BindingDB|TTD
PTPN1 2-(4''-(2-Butylbenzofuran-3-yl)biphenyl-4-yloxy)acetic acid NA 457000000 NA NA NA NA BindingDB