| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN1 |
(2-Butyl-1-benzofuran-3-yl)-(6-hydroxynaphthalen-2-yl)methanone |
NA |
3160000|3162277.66 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
(2R)-2-[4-[4-(3-benzylimidazo[4,5-b]pyridin-2-yl)phenyl]phenoxy]-3-phenylpropanoic acid |
NA |
213000000|213796209 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
4'-(2-Butyl-benzofuran-3-yl)-biphenyl-4-ol |
NA |
741000000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
2-Methoxy-naphthalene-1,6-dicarboxylic acid |
NA |
20000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
2-Methoxy-naphthalene-1,6-dicarboxylic acid 6-methyl ester |
NA |
2800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
2-Hydroxy-naphthalene-1,6-dicarboxylic acid |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
3-(Carboxyformamido)isonicotinic acid |
158489.32|159000|160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
3-Carboxymethoxy-naphthalene-2,7-dicarboxylic acid |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
1-(tert-Butylperoxy)-1,2-benziodoxol-3(1H)-one |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
2-(1-carboxy-N-methylformamido)benzoic acid |
1090000|1096478.2|1100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
2-(Carboxyformamido)-6-methylbenzoic acid |
1698243.65|1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
6-(Carboxy-difluoro-methoxy)-naphthalene-2-carboxylic acid |
NA |
9400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
2-Naphthylglycolic acid |
NA |
3300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
Oxo-pentafluorophenyl-acetic acid |
NA |
790000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
4-Methoxymandelic acid |
NA |
5700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
N-[(3S)-2-[3-(3-chlorophenyl)propanoyl]-3-(methylcarbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfamic acid |
NA |
101100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
N-[(3S)-3-(benzylcarbamoyl)-2-[(tert-butoxy)carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfamic acid |
NA |
120200 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
3-(4-Methoxybenzofuran-5-yl)-5-phenyl-4,5-dihydroisoxazole |
NA |
227000 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
N-[(3S)-2-[3-(4-methoxyphenyl)propanoyl]-3-(methylcarbamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfamic acid |
NA |
242000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
N-[(3S)-3-(methylcarbamoyl)-2-[3-(4-methylphenyl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfamic acid |
NA |
198000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |