| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTGS2 |
5-Chloro-3-(3,4-difluorophenyl)-2-(4-methylsulfonylphenyl)pyran-4-one |
NA |
1234809.61 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTGS2 |
Acetic acid 2-benzylsulfanyl-phenyl ester |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTGS2 |
5-(4-Methanesulfonyl-phenyl)-6-phenyl-thiazolo[3,2-b][1,2,4]triazole |
NA |
10000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTH1R |
2-Cyclohexyl-8-[2-[2,6-dimethyl-4-(2-oxoimidazolidin-1-yl)phenyl]ethylsulfonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| PTH1R |
trans-Sulindac |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Geranyl acetate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Allylthiourea |
NA |
NA |
NA |
NA |
141254 |
NA |
PubChem |
| PTH1R |
Chlorzoxazone |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Ethionamide |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
(1R,4S,5'S,6R,6'R,8R,12S,13S,20R,21R,24S)-6'-[(2S)-butan-2-yl]-21,24-dihydroxy-12-[(2R,4S,5S,6S)-5-[(2S,4S,5S,6S)-5-hydroxy-4-methoxy-6-methyloxan-2-yl]oxy-4-methoxy-6-methyloxan-2-yl]oxy-5',11,13,22-tetramethylspiro[3,7,19-trioxatetracyclo[15.6.1.14,8.020,24]pentacosa-10,14,16,22-tetraene-6,2'-oxane]-2-one |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Ursodiol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Butylated Hydroxytoluene |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Ebselen |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Moricizine Hydrochloride |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Glyburide |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Isomaltose |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Naringenin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Nifenazone |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Butoconazole Nitrate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
8-(3-Chlorophenyl)sulfonyl-2-(2,4-dichlorophenyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |