Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| PTGS2 | 6-Maleimidohexanoic acid | NA | 800000 | NA | NA | NA | NA | TTD |
| PTGS2 | Bz(4-F)-Tyr-Met-Asp-OH | NA | 1000000 | NA | NA | NA | NA | TTD |
| PTGS2 | Bz(4-F)-Phe-Met-Asp-OH | NA | 450000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Bz(4-F)-Tyr-Ser-OH | NA | 140000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Bz(4-F)-Trp-Met-Asp-OH | NA | 450000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | (2S)-2-[[(2S)-2-[(4-fluorobenzoyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]butanedioic acid | NA | 110000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | 2-[1-(4-Chlorobenzoyl)-2-phenylindol-3-yl]acetic acid | NA | 400000 | NA | NA | NA | NA | TTD |
| PTGS2 | (2S)-2-[[(2S)-2-[(4-fluorobenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-hydroxypropanoic acid | NA | 200000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Trp-Tyr-Asp | NA | 700000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Bz(4-F)-Trp-Met-Glu-OH | NA | 350000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Bz(4-F)-Tyr-Met-Glu-OH | NA | 500000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Bz(4-F)-Phe-Met-Glu-OH | NA | 1000000 | NA | NA | NA | NA | TTD |
| PTGS2 | Bz(4-F)-Tyr-Trp-Ser-OH | NA | 180000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
| PTGS2 | Cinnamaldehyde | NA | 245000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| PTGS2 | Trihydroxychalcone | NA | 130000 | NA | NA | NA | NA | BindingDB|TTD |
| PTGS2 | Ursolic Acid | NA | 130000 | NA | NA | NA | NA | BindingDB|PubChem |
| PTGS2 | Carumonam | NA | NA | NA | NA | NA | 500000 | PubChem |
| PTGS2 | Caffeic Acid | NA | 129700 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| PTGS2 | Thymol | NA | NA | NA | NA | NA | 120000 | PubChem |