| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTPN1 |
3-(Carboxymethoxy)-4-methylthiophene-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
3-(Carboxymethoxy)-4-phenylthiophene-2-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
Sodium;5-[difluoro(naphthalen-2-yl)methyl]-1,2,3-triaza-4-azanidacyclopenta-2,5-diene |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
6-Methylnaphthalen-2-ol |
NA |
707000000|707945784.4 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
|
NA |
156600 |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
5-benzyl-3-Bromo-2-hydroxybenzoic acid |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
Diethyl-[2-(4-naphtho[1,2-d]oxazol-2-yl-phenoxy)-ethyl]-amine |
355000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
2-[(5Z)-5-[[3-(2-amino-2-oxoethoxy)-4-methoxyphenyl]methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
NA |
679000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
Benzoic acid, 3,3'-methylenebis[5-bromo-2-hydroxy- |
NA |
149000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
5-Bromo-4-hydroxy-[1,1'-biphenyl]-3-carboxylic acid |
NA |
351000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
Chromocarb |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
3-[(4-Chlorobenzyl)sulfanyl]-2-thiophenecarboxylic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
5-(4-Bromophenyl)isoxazole-3-carboxylic acid |
NA |
NA |
800000|8e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTPN1 |
2-(2-Hydroxy-1,1,1,3,3,3-hexafluoropropyl)-1-naphthol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
4-amino-3-bromo-5-cyano-2-hydroxy-benzoic Acid |
NA |
NA |
910000 |
NA |
NA |
NA |
BindingDB |
| PTPN1 |
4-[Acetyl(6,7,8,9-tetrahydrodibenzofuran-2-yl)sulfamoyl]benzoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PTPN1 |
Disodium naphthalene-2,6-disulphonate |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
| PTPN1 |
Salicylic Acid |
19400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PTPN1 |
fluorescein (acid form) |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PTPN1 |
O-Iodoxybenzoic acid |
NA |
1160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |