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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN1 5-Methanesulfonylamino-naphthalene-2-sulfonic acid NA 29000000 NA NA NA NA BindingDB|TTD
PTPN1 4''-(2-Bromo-acetyl)-biphenyl-2-carboxylic acid 220000 NA NA NA NA NA BindingDB|TTD
PTPN1 2-[(S)-2-(2-{2-[4-(2-Bromo-acetyl)-phenoxy]-acetylamino}-acetylamino)-5-guanidino-pentanoylamino]-5-guanidino-pentanoic acid 760000 NA NA NA NA NA BindingDB|TTD
PTPN1 3-[4-[(2S)-3-[4-(3-hydroxy-2-methoxycarbonylphenoxy)butylamino]-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-oxopropyl]-N-oxaloanilino]propanoic acid 200000 NA NA NA NA NA TTD
PTPN1 Disodium;2-fluoro-2-naphthalen-2-yloxypropanedioate NA 320000 NA NA NA NA TTD
PTPN1 Sodium;2,2-difluoro-2-naphthalen-2-ylacetate NA 640000 NA NA NA NA TTD
PTPN1 Sodium;difluoro(naphthalen-2-yl)methanesulfonate NA 175000 NA NA NA NA TTD
PTPN1 Disodium;2-fluoro-2-(3-phenylphenoxy)propanedioate NA 250000 NA NA NA NA TTD
PTPN1 Sodium;2,2-difluoro-2-(3-phenylphenyl)acetate NA 435000 NA NA NA NA TTD
PTPN1 NA NA 15600000 NA NA NA BindingDB
PTPN1 5-(3-Butyramidophenyl)isoxazole-3-carboxylic acid 125893|148000|125892.54 NA NA NA NA NA BindingDB|TTD
PTPN1 Fluoro{7-[fluoro(phosphonato)methyl]-2-naphthyl}methylphosphonate NA 130000 NA NA NA NA BindingDB
PTPN1 [Fluoro-[7-[fluoro(phosphono)methyl]naphthalen-2-yl]methyl]phosphonic acid NA 130000 NA NA NA NA TTD
PTPN1 Difluoro(1-naphthyl)methylphosphonate NA|255000 112000|NA NA NA NA NA BindingDB
PTPN1 1,4-Diiodyl-benzene NA 1410000 NA NA NA NA BindingDB|TTD
PTPN1 1,3-Dioxo-1H-1lambda*5*-ioda-2,4-dioxa-3lambda*5*-phospha-naphthalene-1,3-diol NA 350000 NA NA NA NA BindingDB|TTD
PTPN1 5-Iodyl-1H-imidazole NA 1050000 NA NA NA NA BindingDB|TTD
PTPN1 methyl 2-[4-[[(2S)-2-acetamido-3-[4-(trifluoromethylsulfonylamino)phenyl]propanoyl]amino]butoxy]-6-hydroxybenzoate 200000 NA NA NA NA NA TTD
PTPN1 methyl 2-[4-[[(2S)-2-acetamido-3-[4-[(2,2,2-trifluoroacetyl)amino]phenyl]propanoyl]amino]butoxy]-6-hydroxybenzoate 200000 NA NA NA NA NA TTD
PTPN1 methyl 2-[4-[[(2S)-2-acetamido-3-[4-[(2-hydroxyacetyl)amino]phenyl]propanoyl]amino]butoxy]-6-hydroxybenzoate 200000 NA NA NA NA NA TTD