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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTPN1 methyl 2-[4-[[(2S)-2-acetamido-3-[4-[(3-hydroxypyridine-2-carbonyl)amino]phenyl]propanoyl]amino]butoxy]-6-hydroxybenzoate 200000 NA NA NA NA NA TTD
PTPN1 2-[4-[(2S)-2-acetamido-3-[4-(3-hydroxy-2-methoxycarbonylphenoxy)butylamino]-3-oxopropyl]-2-aminophenoxy]acetic acid 200000 NA NA NA NA NA TTD
PTPN1 2-(Oxaloamino)thiophene-3-carboxylic acid 107151.93|108000 NA NA NA NA NA BindingDB|TTD
PTPN1 Hydrogen (2-naphthyloxy)methylphosphonate 1300000 NA NA NA NA NA BindingDB
PTPN1 Naphthalen-2-yloxymethylphosphonic acid 1300000 NA NA NA NA NA TTD
PTPN1 Dioxido-oxo-(phenoxymethyl)-lambda5-phosphane 3300000 NA NA NA NA NA BindingDB
PTPN1 Hydrogen (1-phenanthryloxy)methylphosphonate 410000 NA NA NA NA NA BindingDB
PTPN1 Phenanthren-1-yloxymethylphosphonic acid 410000 NA NA NA NA NA TTD
PTPN1 Hydrogen (1-naphthyloxy)methylphosphonate 1300000 NA NA NA NA NA BindingDB
PTPN1 Naphthalen-1-yloxymethylphosphonic acid 1300000 NA NA NA NA NA TTD
PTPN1 [4-(Carboxymethyl)phenoxy]methylphosphonate 1100000 NA NA NA NA NA BindingDB
PTPN1 [4-(Phosphonomethoxy)phenyl]acetic acid 1100000 NA NA NA NA NA TTD
PTPN1 2-[4-[4-(2-Benzylthiophen-3-yl)phenyl]phenoxy]acetic acid NA 83100000|83176377.11 NA NA NA NA BindingDB|TTD
PTPN1 2-Butyl-3-(phenylmethyl)benzofuran NA 691000000|691830970.9 NA NA NA NA BindingDB|TTD
PTPN1 2-[4-(4-Methylphenyl)-2-phenylphenoxy]acetic acid NA 46700000|46773514.13 NA NA NA NA BindingDB|TTD
PTPN1 2-Butyl-3-methyl-1-benzofuran NA 707000000|707945784.4 NA NA NA NA BindingDB|TTD
PTPN1 2-[4-[4-(2-Benzyl-1-benzothiophen-3-yl)phenyl]phenoxy]acetic acid NA 70700000|70794578.44 NA NA NA NA BindingDB|TTD
PTPN1 2-[4-[4-(2-Ethyl-1-benzothiophen-3-yl)phenyl]phenoxy]acetic acid NA 89100000|89125093.81 NA NA NA NA BindingDB|TTD
PTPN1 2-[2-(4-Methoxyphenyl)-4-(4-methylphenyl)phenoxy]acetic acid NA 46700000|46773514.13 NA NA NA NA BindingDB|TTD
PTPN1 [Difluoro-(3-phenylethynyl-phenyl)-methyl]-phosphonic acid NA 135900 NA NA NA NA BindingDB|TTD