| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RNASE1 |
3'-O-Acetylthymidine |
NA |
197000 |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
Cytidine 3'-monophosphate |
NA|103000 |
312000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
2-amino-N-[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]-3-(4-hydroxyphenyl)propanamide |
451000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
2-[[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-2-oxoacetic acid |
132000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
3-[[(2S,3R,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxopyrimidin-1-yl)oxolan-3-yl]amino]-3-oxopropanoic acid |
380000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
1-[3-(4-Carboxypiperidin-1-YL)-3-deoxy-beta-D-arabinofuranosyl]pyrimidine-2,4(1H,3H)-dione |
103000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASEL |
Vitexin |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| RNASEL |
Myricetin |
NA |
264000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| RNASEL |
Butylparaben |
NA |
2400000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|PubChem |
| RNMT |
N-[[(2R,3S,4R,5R)-5-[4-amino-5-(2-quinolin-3-ylethynyl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-dihydroxyoxolan-2-yl]methyl]-3-cyano-4-methoxy-N-methylbenzenesulfonamide |
NA |
165300 |
NA |
NA |
NA |
NA |
BindingDB |
| RNPEP |
(5S)-5-amino-2,7-dimethyl-4-oxooctanoic acid |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RNPEP |
3-Amino-2-hydroxy-5-methyl-hexanoic acid (3-methyl-butyl)-amide |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| RNPEP |
(3S)-3-amino-5-methylhexan-2-one |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| RNPEP |
Ubenimex |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| ROCK1 |
3-(4-Methyl-1,4-diazepan-1-yl)-5-(3-methylpyridin-4-yl)pyrazin-2-amine |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ROCK1 |
5-bromo-N-(pyridin-4-yl)nicotinamide |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| ROCK1 |
1-(1H-indazol-5-yl)-3-phenylurea |
NA |
157100 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| ROCK1 |
5-(4-fluorophenyl)-N-pyridin-4-ylpyridine-3-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK1 |
4-(4-fluorophenyl)-N-pyridin-4-ylpyridine-3-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| ROCK1 |
5-Aminoindazole |
NA |
181300 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |