| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RIR |
(2S)-2-[[(2S)-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-[[2-benzyl-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylbutanoyl]amino]-3-methylbutanoyl]amino]-4-oxobutanoyl]amino]-3-carboxypropanoyl]amino]-4-methylpentanoic acid |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Phe-Leu-Asp-Ala-Asp-Phe-OH |
NA |
412000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Leu-Asp-Ala-Asp-Phe-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
2-[3-Carboxy-2-(2-{3-methyl-2-[2-(3-phenyl-propionylamino)-acetylamino]-butyrylamino}-4-oxo-4-pyrrolidin-1-yl-butyrylamino)-propionylamino]-4-methyl-pentanoic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
1-[[2-(2-{2-[(2-Benzyl-3-phenyl-propionyl)-methyl-amino]-3-methyl-butyrylamino}-3,3-dimethyl-butyrylamino)-3-carbamoyl-propionylamino]-(1-hydroxymethyl-3,3-dimethyl-butylcarbamoyl)-methyl]-cyclopentanecarboxylic acid |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| RIR |
Val-Val-Asn-Asp-Leu |
NA |
760000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Leu-aThr-Leu-Asp-Ala-Asp-Phe-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-aThr-Leu-Asp-Ala-Asp-Phe-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
H-Phe-aThr-Leu-Asp-Ala-Asp-Phe-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Phe-aThr-Leu-Asp-Ala-Asp-Phe-Ala-Ala-OH |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Phe-aThr-Leu-Asp-Ala-Asp-Leu-OH |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Phe-aThr-Leu-Asp-Asp-Phe-OH |
NA |
322000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
Ac-Phe-aThr-Ala-Asp-Ala-Asp-Phe-OH |
NA |
207000 |
NA |
NA |
NA |
NA |
TTD |
| RIR |
1-Aminoadenosine |
NA |
232000 |
NA |
NA |
NA |
NA |
TTD |
| RNASE1 |
Thymidine, 3'-benzoate |
NA |
341000 |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
3'-Thymidylic acid |
NA |
167000 |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
2-((2S,3S,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3-ylamino)-2-oxoacetic acid |
132000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
3-((2S,3S,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3-ylamino)-3-oxopropanoic acid |
380000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
4-((2S,3S,5R)-2-(hydroxymethyl)-5-(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-3-ylamino)-4-oxobutanoic acid |
918000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RNASE1 |
3''-[1-(4-Ethoxycarbonylpiperdinyl)]-3''-deoxy-ara-uridine |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |