| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
6-Chloro-4-(4-chlorophenyl)sulfanyl-1-methylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(5-chloro-4-phenylmethoxy-1H-benzimidazol-2-yl)acetonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
1-methyl-N-piperidin-3-ylindol-4-amine |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-(2-phenylethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1S,2R)-2-[[5,6-dichloro-1-[(2,5-dichlorophenyl)methyl]-2-(hydroxymethyl)benzimidazol-4-yl]oxymethyl]cyclohexan-1-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-pyridin-2-ylsulfanyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1-Benzyl-6-chloro-5-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
7-[[6-chloro-2-(hydroxymethyl)-1H-indol-4-yl]oxy]-3,4-dihydro-1H-quinolin-2-one |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
N-[(1-benzylpyrrolidin-3-yl)methyl]-6-chloro-4-(4-chlorophenyl)sulfanyl-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[4-bromo-2-cyano-6-(3,4-dichlorophenyl)sulfanylindol-1-yl]methyl]-N,N-dimethylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-6-[(4-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-[2-(3-methoxyphenyl)ethyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1S,2R)-2-[[5,6-dichloro-2-(hydroxymethyl)-1-methylbenzimidazol-4-yl]oxymethyl]cyclohexan-1-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-4-(4-chlorophenyl)sulfanyl-1-methylindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[(6-aminopyridin-2-yl)methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]-1H-pyrimidin-6-one |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-bromo-6-phenoxy-1-[[4-(2H-tetrazol-5-yl)phenyl]methyl]indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-(2-indol-1-ylethyl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(4-Aminophenyl)-5,6-dichloro benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-(pyrrolidin-2-ylmethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |