| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
4-(2-Chlorophenoxy)-1-methylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-Chloro-6-phenylmethoxy-1-propylbenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-6-(3,4-dichlorophenyl)sulfanyl-1-[[4-(propan-2-ylcarbamoyl)phenyl]methyl]indole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6,7-dichloro-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)-3H-benzimidazole-5-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
methyl 4-(4-chlorophenyl)sulfanyl-1H-indole-6-carboxylate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1S,2R)-2-[[5,6-dichloro-2-(hydroxymethyl)-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-4-yl]oxymethyl]cyclohexan-1-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-bromo-6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-4-(cyclohexylmethoxy)-2-ethenyl-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(3-Fluorophenoxy)-1-methylindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(7-Chloro-1-ethyl-5-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1-Ethyl-5-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(2-Chlorophenoxy)-1-methylindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]benzonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-1-[[4-[4-[(2-methylpropan-2-yl)oxycarbonyl]piperazine-1-carbonyl]phenyl]methyl]-6-phenoxyindole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-(pyrrolidin-3-ylmethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
Tert-butyl 4-[[4-bromo-2-(hydroxymethyl)-6-phenoxyindol-1-yl]methyl]benzoate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-(Benzyloxy)-1-ethyl-1H-benzo[d]imidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-(2-methylsulfonylethyl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(3-chlorophenoxy)-1H-indol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |