| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
[5-Chloro-6-[(2-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
1-(6-chloro-4-phenoxy-1H-indol-2-yl)ethanone |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-4-(4-chlorophenyl)sulfanyl-1H-indol-2-yl]-(4-methylpiperazin-1-yl)methanone |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-2-[4-(2H-tetrazol-5-yl)phenyl]-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1-Methyl-4-phenoxyindol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6,7-dichloro-4-(2,4-dichlorophenyl)sulfanyl-N-(1-methylazetidin-3-yl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(4-phenoxy-1H-benzimidazol-2-yl)acetonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[(4-aminopyrimidin-2-yl)methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4,5-dichloro-6-[(4-methoxyphenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-6-[(3,4-dichlorophenyl)methylsulfanyl]-1-[[4-(dimethylcarbamoyl)phenyl]methyl]indole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(2,6-dichlorophenoxy)-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-Chloro-4-(4-chlorophenyl)sulfanyl-1-pyridin-3-ylsulfonylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-bromo-6-(3,4-dichlorophenyl)sulfanyl-N-[[(2S)-1-methylpyrrolidin-2-yl]methyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(4-cyclohexyl-6-phenoxy-1H-indol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5-chloro-4-(4-chlorophenyl)sulfanyl-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzimidazol-1-yl]acetic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-phenoxy-4-piperidin-3-yl-1H-indol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(1H-indol-4-ylsulfanyl)-N-methylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-2-[3-(4-methylpiperazin-1-yl)phenyl]-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-(4-chlorophenyl)sulfanyl-1-(1H-1,2,4-triazol-5-ylmethyl)indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5,6-dichloro-1-[[3-(2H-tetrazol-5-yl)phenyl]methyl]benzimidazol-2-yl]-1,3-oxazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |