| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
[6-chloro-5-[(2-fluorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-4-(cyclohexylmethoxy)-2-pyridin-4-yl-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[[4-Bromo-2-(hydroxymethyl)-6-phenoxyindol-1-yl]methyl]phenyl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]benzonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-bromo-1-[[4-(dimethylcarbamoyl)phenyl]methyl]-N-[(1-methylpiperidin-4-yl)methyl]-6-naphthalen-2-ylsulfanylindole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(1H-indol-4-ylsulfanyl)benzoic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(3,5-dichlorophenyl)-N-(1-methylazetidin-3-yl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1-Benzyl-5-chloro-6-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-4-(2-phenylethoxy)-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-chloro-6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-(1H-imidazol-2-yl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(4-phenoxy-1H-indol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-4-(4-chlorophenyl)sulfanyl-1H-indol-2-yl]-(4-methyl-1,4-diazepan-1-yl)methanone |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(4-chlorophenyl)-(1H-indol-4-yl)methanone |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(4-chlorophenoxy)-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(3R,4S)-3-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]piperidin-4-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(1H-indol-4-ylsulfanyl)benzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(6-chloro-5-phenylmethoxy-1H-benzimidazol-2-yl)acetonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
Tert-butyl 4-[[4-bromo-6-(3,4-dichlorophenyl)sulfanyl-2-[2-(1-methylpiperidin-4-yl)ethylcarbamoyl]indol-1-yl]methyl]benzoate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-5-[(4-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |