| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
1-[6-chloro-4-(4-chlorophenyl)sulfanyl-1H-indole-2-carbonyl]piperidine-3-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-(oxan-4-ylmethyl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4,6-bis[(4-chlorophenyl)sulfanyl]-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[4-bromo-6-(3,4-dichlorophenyl)sulfanyl-2-[(dimethylamino)methyl]indol-1-yl]methyl]-N,N-dimethylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-Chloro-1-ethyl-6-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-(benzenesulfinyl)-4-bromo-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-1-[2-(4-carboxyphenyl)ethyl]-6-phenoxyindole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-2-(2-piperazin-1-ylpyridin-4-yl)-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzoic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[4-bromo-6-(3,4-dichlorophenyl)sulfanyl-2-(methylaminomethyl)indol-1-yl]methyl]-N,N-dimethylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-2-(4-pyridin-4-ylphenyl)-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(4-Fluorophenoxy)-1-methylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(1-Benzyl-5,6-dichlorobenzimidazol-2-yl)-1,2,5-oxadiazol-3-amine |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-5-[(3-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-chlorophenyl)sulfonyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-1-ethyl-5-[(2-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1-Benzyl-4-bromo-6-phenylmethoxyindol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[(3,4-dichlorophenyl)methylsulfanyl]-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-methyl-6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |