| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
5-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]pyrrolidin-2-one |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-1-ethyl-5-[(4-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-5-phenylmethoxy-1-(2,2,2-trifluoroethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-6-(3,4-dichlorophenyl)sulfanyl-1-[[4-[4-[(2-methylpropan-2-yl)oxycarbonyl]piperazine-1-carbonyl]phenyl]methyl]indole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-chlorophenyl)sulfinyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-6-[(3-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-1-ethyl-6-[(3-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6,7-dichloro-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)-3H-benzimidazol-5-yl]-(4-methylpiperazin-1-yl)methanone |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
tert-butyl N-[[4,5-dichloro-6-[(4-chlorophenyl)methoxy]-1H-benzimidazol-2-yl]methyl]carbamate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
methyl 4-(1H-indol-4-ylsulfanyl)benzoate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-6-phenylmethoxy-1-(2,2,2-trifluoroethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(4-Chlorophenoxy)-1-methylindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(4-chlorophenyl)sulfanyl-N-[(5-oxopyrrolidin-2-yl)methyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-(cyclopent-3-en-1-ylmethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-1-[[4-[(1-methylpyrrolidin-3-yl)carbamoyl]phenyl]methyl]-6-phenoxyindole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(2-Fluorophenoxy)-1-methylindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzoic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-6-(3,4-dichlorophenyl)sulfanyl-1-[[4-(piperazine-1-carbonyl)phenyl]methyl]indole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |