| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
[4-[[(1S,2R)-2-aminocyclohexyl]methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-bromo-4,5-dichloro-2-pyridin-4-yl-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]oxolan-3-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-chloro-6-phenylmethoxy-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(5,6-dichloro-1H-benzimidazol-2-yl)-N-[[(2S)-1-methylpyrrolidin-2-yl]methyl]benzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[1-(2-Aminoethyl)-6-chloro-4-phenoxyindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(1-methylpyrazol-3-yl)-6-phenoxy-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(3,5-dichlorophenyl)-N-[2-(1-methylpiperidin-4-yl)ethyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-chloro-1-(1H-imidazol-5-ylmethyl)-6-phenoxyindol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[(4-aminopyrimidin-5-yl)methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
tert-butyl 4-[4-(5,6-dichloro-1H-benzimidazol-2-yl)pyridin-2-yl]piperazine-1-carboxylate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-4-(3,4-dimethoxyphenyl)sulfanyl-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
7-Chloro-2-(ethoxymethyl)-1-ethyl-5-phenylmethoxybenzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-methoxyphenyl)sulfanyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
methyl 4-(4-bromophenyl)sulfanyl-6-chloro-1H-indole-2-carboxylate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-[2-(1H-imidazol-5-yl)ethoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(5-chloro-4-phenoxy-1H-benzimidazol-2-yl)-1,3-oxazole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
Tert-butyl 4-[(4-bromo-6-phenoxyindol-1-yl)methyl]benzoate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(4-chlorophenyl)sulfanyl-1H-indole-6-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-Chloro-5-phenylmethoxy-1-propylbenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |