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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
RHEB [4-(4-Fluorophenoxy)-1-methylindol-2-yl]methanol NA 550000 NA NA NA NA BindingDB
RHEB 6-chloro-4-(4-chlorophenyl)sulfanyl-N-(1-methylpiperidin-4-yl)-1H-indole-2-carboxamide NA 550000 NA NA NA NA BindingDB
RHEB (6-Chloro-1-methyl-4-phenoxyindol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (3R,4R)-3-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]piperidin-4-ol NA 550000 NA NA NA NA BindingDB
RHEB [4-[(2-aminopyridin-3-yl)methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol NA 550000 NA NA NA NA BindingDB
RHEB 5-Chloro-1-ethyl-6-phenylmethoxybenzimidazole NA 550000 NA NA NA NA BindingDB
RHEB (6-phenoxy-4-piperidin-4-yl-1H-indol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (1,4-Dimethyl-6-phenoxyindol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (6-Chloro-1-ethyl-5-phenoxybenzimidazol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (4-methyl-6-phenoxy-1H-indol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB [6-(benzenesulfonyl)-4-bromo-1H-indol-2-yl]methanol NA 550000 NA NA NA NA BindingDB
RHEB 4-(3,4-dichlorophenyl)sulfanyl-1H-indole NA 550000 NA NA NA NA BindingDB
RHEB 4-Chloro-2-(ethoxymethyl)-1-ethyl-6-phenylmethoxybenzimidazole NA 550000 NA NA NA NA BindingDB
RHEB 4-(4-Chlorophenyl)sulfanyl-1-methylindole NA 550000 NA NA NA NA BindingDB
RHEB (6-chloro-4-phenylmethoxy-1H-benzimidazol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB 4-(5,6-dichloro-1H-benzimidazol-2-yl)-N-[2-(1-methylpiperidin-4-yl)ethyl]benzamide NA 550000 NA NA NA NA BindingDB
RHEB [4-(3-fluorophenoxy)-1H-indol-2-yl]methanol NA 550000 NA NA NA NA BindingDB
RHEB (6-chloro-4-phenoxy-1H-benzimidazol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (6-chloro-4-phenylmethoxy-1H-indol-2-yl)methanol NA 550000 NA NA NA NA BindingDB
RHEB (4-Chloro-1-ethyl-6-phenylmethoxybenzimidazol-2-yl)methanol NA 550000 NA NA NA NA BindingDB