| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
(6-phenoxy-1H-indol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(4-fluorophenoxy)-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(4-chlorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-Chloro-1-methyl-6-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-chloro-4-phenoxy-1H-benzimidazol-2-yl)methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-(oxolan-2-ylmethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(4-fluorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]piperidin-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-Chloro-1-ethyl-5-phenylmethoxybenzimidazole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(2,4-dichlorophenyl)methylsulfanyl]-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(3-chlorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(3-fluorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5,6-dichloro-1-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzimidazol-2-yl]-1,3-oxazole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]cyclopentan-1-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(5,6-Dichloro-1H-benzimidazol-2-yl)-1,2,5-oxadiazol-3-amine |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(2-chlorophenoxy)-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-[(2-chloropyrimidin-4-yl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-5-[(2-chlorophenyl)methoxy]-1-ethylbenzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(4-chlorophenyl)sulfanyl-2-methyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-Fluorophenoxy)-1-methylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |