| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
6-chloro-4-(2,4-dichlorophenyl)sulfanyl-N-(1-methylpiperidin-4-yl)-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-Chloro-1-ethyl-5-phenylmethoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-bromo-6-(3,4-dichlorophenyl)sulfanyl-N-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(5-chloro-4-phenoxy-1H-indol-2-yl)ethyl acetate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[4-bromo-6-(3,4-dichlorophenyl)sulfanyl-2-(methoxymethyl)indol-1-yl]methyl]-N,N-dimethylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(2-chlorophenyl)sulfinyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-1-ethyl-6-[(4-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-bromo-6-(3,4-dichlorophenyl)sulfanyl-N-[2-(1-methylpiperidin-4-yl)ethyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5-chloro-1-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzimidazol-2-yl]-1,3-oxazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(1R,2R)-2-[[5,6-dichloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]cyclohexan-1-ol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(4-chlorophenyl)sulfonyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(4-phenoxy-1H-benzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-1-[[4-(dimethylcarbamoyl)phenyl]methyl]-6-[4-(trifluoromethyl)phenyl]sulfanylindole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(2-chlorophenyl)sulfonyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
1-[(4-Bromophenyl)methyl]-6-chloro-4-(2,4-dichlorophenyl)sulfanylindole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-2-(2-phenylpyridin-4-yl)-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-(5-chloro-4-phenoxy-1H-benzimidazol-2-yl)acetonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
7-(4-chlorophenyl)sulfanyl-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5-chloro-6-phenoxy-1H-indole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |