| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
[4-(1-methylpyrazol-4-yl)-6-phenoxy-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-Chlorophenoxy)-1-methylindole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-Chloro-1-methyl-4-phenoxyindol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[(2-aminopyrimidin-4-yl)methoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[2-(aminomethyl)-4-bromo-6-(3,4-dichlorophenyl)sulfanylindol-1-yl]methyl]-N,N-dimethylbenzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-Chloro-1-ethyl-6-phenoxybenzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5,6-dichloro-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzimidazol-1-yl]acetic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(1H-indol-4-ylsulfanyl)phenyl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(5,6-dichloro-1H-benzimidazol-2-yl)-N,N-dimethylpyridin-2-amine |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-Chloro-1-methyl-4-phenylmethoxyindol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5-Chloro-1-ethyl-6-[(2-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6,7-dichloro-4-(2,4-dichlorophenyl)sulfanyl-N-[2-(1-methylpiperidin-4-yl)ethyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[7-phenoxy-1-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzimidazol-2-yl]-1,3-oxazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-Bromo-6-phenoxy-1-[[4-(piperazine-1-carbonyl)phenyl]methyl]indole-2-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(5,6-dichloro-1H-benzimidazol-2-yl)-N-[[(2R)-1-methylpyrrolidin-2-yl]methyl]benzamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-Chloro-1-ethyl-5-[(3-fluorophenyl)methoxy]benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-bromo-6-phenoxy-1-(1H-1,2,4-triazol-5-ylmethyl)indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[5,6-dichloro-4-(piperidin-2-ylmethoxy)-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(2,4-dichlorophenyl)sulfanyl-N-[2-(4-phenylpiperazin-1-yl)ethyl]-1H-indole-2-carboxamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-[(2-chlorophenyl)methoxy]-1H-benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |