| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| REN |
2-{2-[2-(2-Hydroxy-3-methyl-butyrylamino)-4-methyl-pentanoylamino]-3-methyl-butyrylamino}-3-phenyl-propionic acid methyl ester |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-hydroxy-2-phenylacetyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate |
980000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| REN |
methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-hydroxy-2-phenylacetyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate |
530000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| REN |
methyl (2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-hydroxy-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate |
670000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| REN |
methyl (2S)-2-[[(2S)-2-[[5-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxy-7-methyloctanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate;dihydrochloride |
900000|3000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
methyl (2R)-2-[[(2R)-2-[[5-[[(2S)-2-amino-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxy-7-methyloctanoyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoate;dihydrochloride |
740000|1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| REN |
H-His-Leu-Leu-Val-Phe-OMe.2HCl |
540000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RGS8 |
2,4-Dibutyl-1,2,4-thiadiazolidine-3,5-dione |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RGS8 |
4-[(4-Methoxyphenyl)methyl]-2-(4-methylphenyl)-1,2,4-thiadiazolidine-3,5-dione |
NA |
312000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RGS8 |
4-Butyl-2-tert-butyl-1,2,4-thiadiazolidine-3,5-dione |
NA |
119000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RGS8 |
2-Tert-butyl-4-(2-methylpropyl)-1,2,4-thiadiazolidine-3,5-dione |
NA |
194000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RHEB |
5,6-Dichloro-2-(4-(4-methylpiperazin-1-yl)phenyl)-1H-benzo[d]imidazole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-isoquinolin-5-yloxy-1H-indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
1-methyl-N-piperidin-4-ylindol-4-amine |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[[6-chloro-2-(hydroxymethyl)-1H-benzimidazol-4-yl]oxymethyl]cyclohexan-1-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-(3,4-dimethoxyphenyl)sulfanyl-1H-indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(4-bromo-6-phenoxy-1H-benzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
5,6-dichloro-4-[(4-chlorophenyl)methoxy]-2-methyl-1H-benzimidazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[4-(2,4-Dichlorophenyl)sulfanylindol-1-yl]methyl]benzonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(5-chloro-4-phenoxy-1H-indol-2-yl)methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |