| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RHEB |
2-[6-Chloro-2-(hydroxymethyl)-5-phenylmethoxybenzimidazol-1-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
Tert-butyl 4-[(5,6-dichloro-2-pyridin-4-ylbenzimidazol-1-yl)methyl]benzoate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
1-(Carboxymethyl)-6-chloro-4-(2,5-dichlorophenoxy)indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(2-fluorophenoxy)-1H-indol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[6-chloro-5-phenylmethoxy-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-(5-chloro-4-phenoxy-1H-indol-2-yl)propanoic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-[2-(2-aminopyridin-4-yl)ethoxy]-5,6-dichloro-1H-benzimidazol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[2-[5,6-dichloro-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)benzimidazol-1-yl]ethyl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(2-chlorophenoxy)-1-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-yl]methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
3-[5,6-dichloro-1-[[4-(2H-tetrazol-5-yl)phenyl]methyl]benzimidazol-2-yl]-1,2,5-oxadiazole |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(2-fluorophenoxy)-1H-indole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-phenoxy-1H-indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-[[5,6-Dichloro-2-(1,3-oxazol-2-yl)benzimidazol-1-yl]methyl]benzonitrile |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-phenyl-1H-indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
6-chloro-4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]-1H-indole-2-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
(6-chloro-5-phenylmethoxy-1H-benzimidazol-2-yl)methanol |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
Methyl 1-[(4-bromophenyl)methyl]-6-chloro-4-(2,4-dichlorophenyl)sulfanylindole-2-carboxylate |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
[4-(2-chlorophenoxy)-1H-indol-2-yl]methanol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
4-(3-fluorophenoxy)-1H-indole |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| RHEB |
2-[5-Chloro-2-(hydroxymethyl)-6-phenylmethoxybenzimidazol-1-yl]acetamide |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |