| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SELE |
(2R)-2-[[2-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetyl]amino]pentanedioic acid |
NA |
7000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
Sodium;3,5-dihydroxy-2-[5-hydroxy-2-(hydroxymethyl)-4-(3,4,5-trihydroxy-6-methyloxan-2-yl)oxyoxan-3-yl]oxy-6-(hydroxymethyl)oxane-4-sulfonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SELE |
2-{[1-(Methoxycarbonylmethyl-carbamoyl)-ethyl]-[2-(3,4,5-trihydroxy-6-phenoxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
3400000|2800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{[1-(Methoxycarbonylmethyl-carbamoyl)-ethyl]-[2-(3,4,5-trihydroxy-6-{3-[4-(4-phenoxy-phenoxy)-phenyl]-propoxymethyl}-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
420000|3420000|3620000|600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{[1-(Methoxycarbonylmethyl-carbamoyl)-ethyl]-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{{2-[6-(4-{2-[2-(2-Ethoxy-ethoxy)-ethoxy]-ethoxy}-butoxymethyl)-3,4,5-trihydroxy-tetrahydro-pyran-2-yl]-acetyl}-[1-(methoxycarbonylmethyl-carbamoyl)-ethyl]-amino}-pentanedioic acid |
NA |
500000|300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{[3-Carboxy-1-(carboxymethyl-carbamoyl)-propyl]-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{[3-Carboxy-1-(methoxycarbonylmethyl-carbamoyl)-propyl]-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{(1-tert-Butylcarbamoyl-ethyl)-[2-(3,4,5-trihydroxy-6-phenoxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
2500000 |
NA |
NA |
NA |
NA |
TTD |
| SELE |
2-{(1-Phenethylcarbamoyl-ethyl)-[2-(3,4,5-trihydroxy-6-phenoxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
2500000 |
NA |
NA |
NA |
NA |
TTD |
| SELE |
2-[[1-(Carboxymethyl-carbamoyl)-2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-ethyl]-(3-carboxy-propionyl)-amino]-pentanedioic acid |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
| SELE |
2-[[1-(Methoxycarbonylmethyl-carbamoyl)-2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-ethyl]-(3-methoxycarbonyl-propionyl)-amino]-pentanedioic acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
N-(1-{Benzyl-[1-(methoxycarbonylmethyl-carbamoyl)-2-(3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yl)-ethyl]-carbamoyl}-2,3-dihydroxy-propyl)-succinamic acid |
NA |
840000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-[2-([1-Phenethylcarbamoyl-2-(3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yl)-ethyl]-{3-[4-(4-phenoxy-phenoxy)-phenyl]-propionyl}-amino)-acetylamino]-pentanedioic acid |
NA |
530000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-(2-{{1-Phenethylcarbamoyl-3-[4-(4-phenoxy-phenoxy)-phenyl]-propyl}-[2-(3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-acetylamino)-pentanedioic acid |
NA |
950000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-[2-(3,4,5-Trihydroxy-6-{3-[4-(4-phenoxy-phenoxy)-phenyl]-propoxymethyl}-tetrahydro-pyran-2-yl)-acetylamino]-pentanedioic acid |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
2-{2-[6-(4-{2-[2-(2-Ethoxy-ethoxy)-ethoxy]-ethoxy}-butoxymethyl)-3,4,5-trihydroxy-tetrahydro-pyran-2-yl]-acetylamino}-pentanedioic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| SELE |
5-[(2R,4S)-2-[[(2S,3R)-1-[2-[2-[2-[[(2S)-1,5-dihexadecoxy-1,5-dioxopentan-2-yl]amino]ethoxy]ethoxy]ethylamino]-1-oxo-3-[(2R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxybutan-2-yl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-5-oxopentanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
5-[(2R,4S)-2-[[(2S,3R)-1-[[2-[[(2S)-1,5-dihexadecoxy-1,5-dioxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-[(2R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxybutan-2-yl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-5-oxopentanoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELE |
5-{(2S,4S)-2-[(1S,2R)-1-Ethoxycarbonyl-2-((2R,5S,6S)-3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yloxy)-propylcarbamoyl]-4-hydroxy-pyrrolidin-1-yl}-5-oxo-pentanoic acid anion |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |