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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
USP7 US10766903, Example 190 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 131 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 195 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 196 NA 100500 NA NA NA NA BindingDB
USP7 6-benzyl-3-[[4-hydroxy-1-[(3R)-3-phenylbutanoyl]piperidin-4-yl]methyl]pyrimidin-4-one NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 197 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 183 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 191 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 237 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 243 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 245 NA 100500 NA NA NA NA BindingDB
USP7 4-(3-Pyrrolidin-3-yl-1,2,4-oxadiazol-5-yl)phenol NA 132000 NA NA NA NA BindingDB|TTD
USP7 2-Amino-3,5-bis(4-hydroxyphenyl)pyridine-4-carbonitrile NA 200000 NA NA NA NA TTD
USP7 4-[3-(1-Methylpyrrolidin-3-yl)-1,2,4-oxadiazol-5-yl]phenol NA 131000 NA NA NA NA BindingDB|TTD
USP7 US10766903, Example 101 NA 100500 NA NA NA NA BindingDB
USP7 (R)-3-((4-Hydroxy-1-(3-phenylbutanoyl)piperidin-4-yl)methyl)-6-((2-methoxyethyl)amino)pyrimidin-4(3H)-one NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 15 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 55 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 135 NA 100500 NA NA NA NA BindingDB
USP7 US10766903, Example 84 NA 100500 NA NA NA NA BindingDB