Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
USP7 | US10766903, Example 190 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 131 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 195 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 196 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | 6-benzyl-3-[[4-hydroxy-1-[(3R)-3-phenylbutanoyl]piperidin-4-yl]methyl]pyrimidin-4-one | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 197 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 183 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 191 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 237 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 243 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 245 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | 4-(3-Pyrrolidin-3-yl-1,2,4-oxadiazol-5-yl)phenol | NA | 132000 | NA | NA | NA | NA | BindingDB|TTD |
USP7 | 2-Amino-3,5-bis(4-hydroxyphenyl)pyridine-4-carbonitrile | NA | 200000 | NA | NA | NA | NA | TTD |
USP7 | 4-[3-(1-Methylpyrrolidin-3-yl)-1,2,4-oxadiazol-5-yl]phenol | NA | 131000 | NA | NA | NA | NA | BindingDB|TTD |
USP7 | US10766903, Example 101 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | (R)-3-((4-Hydroxy-1-(3-phenylbutanoyl)piperidin-4-yl)methyl)-6-((2-methoxyethyl)amino)pyrimidin-4(3H)-one | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 15 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 55 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 135 | NA | 100500 | NA | NA | NA | NA | BindingDB |
USP7 | US10766903, Example 84 | NA | 100500 | NA | NA | NA | NA | BindingDB |