| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
Cianidanol |
NA |
125000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| F2 |
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-methyl-2-oxo-1,3-thiazol-3-yl)acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[(E)-1-[4-[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]ethylideneamino]guanidine |
786000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[4-Carbamimidoyl-2-[2-[(1-pyridin-4-ylpiperidine-4-carbonyl)amino]ethoxy]phenyl]propanoic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[[4-(diaminomethylideneamino)phenyl]methyl]-4-[8-[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazin-1-yl]-8-oxooctanoyl]piperazine-1-carboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Carbamimidoyl-N-[2-(3-carbamimidoyl-phenoxy)-ethyl]-benzamide |
710000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(2,6-Difluorophenyl)pyrido[3,4-d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[(4-Aminomethyl-benzylcarbamoyl)-methyl]-carbamic acid 4-[(4-aminomethyl-benzylcarbamoyl)-methylcarbamoyloxymethyl]-benzyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate |
435000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
1-Methyl-6-(2-methylphenyl)pyrazolo[3,4-d][1,3]oxazin-4-one |
NA |
129000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
7-Ethylsulfanyl-2-(2-fluorophenyl)pyrimido[4,5-d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3aalpha,6aalpha)-3beta,6beta-Bis[4-(4-guanidinobenzylcarbamoyl)piperazinocarbonyloxy]hexahydrofuro[3,2-b]furan |
138000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(2,6-Difluorophenyl)-7-(trifluoromethyl)-4H-3,1-benzoxazine-4-one |
NA |
134000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-piperidin-4-yloxy]-benzoylamino}-ethoxy)-phenyl]-propionic acid |
1500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-amino-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-oxoethyl]-3-hydroxypropanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-Amino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2''-Sulfamoyl-biphenyl-4-carboxylic acid [2-(3-carbamimidoyl-phenoxy)-ethyl]-amide |
NA |
321000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-(7-Carbamimidoyl-naphthalen-2-yl)-2-[4-((S)-pyrrolidin-3-yloxy)-phenyl]-propionic acid |
NA |
1600000 |
NA |
NA |
NA |
NA |
TTD |
| F2R |
H-Ser-Phe-Leu-Leu-D-Arg-NH2 |
NA |
NA |
NA |
109300 |
NA |
NA |
TTD |
| F2R |
deamino-Dab-Phe-Leu-Leu-Arg-NH2 |
NA |
NA |
NA |
730000 |
NA |
NA |
TTD |