| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[3-[(2,5-dihydroxybenzoyl)amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
3542000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
1887000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-5-amino-2-[(2,5-dihydroxybenzoyl)amino]-5-oxopentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2545000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3R)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxybutanoyl]amino]butanoic acid |
NA |
394000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[4-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]butanoylamino]butanoic acid |
NA |
262000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-4-amino-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-4-oxobutanoyl]amino]butanoic acid |
NA |
341000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
((S)-4-Amino-1-{[(1-formyl-4-guanidino-butylcarbamoyl)-methyl]-carbamoyl}-butyl)-carbamic acid tert-butyl ester |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2576000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2R)-2-[(2,5-dihydroxybenzoyl)amino]propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2956000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[6-[(2,5-dihydroxybenzoyl)amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2164000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]acetyl]amino]butanoic acid |
NA |
446000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S,3S)-2-[(2,5-dihydroxybenzoyl)amino]-3-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2710000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-hydroxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2328000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3S)-4-[(2S)-2-[[(2S,3S)-1-[[(1S)-1-carboxypropyl]amino]-3-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-[(2,5-dihydroxybenzoyl)amino]-4-oxobutanoic acid |
NA |
2462000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2R,3S)-2-amino-N-[(2S)-1-[6-aminohexyl-(4-oxothian-3-yl)amino]-1-oxo-3-phenylpropan-2-yl]-3-methylpentanamide |
720000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-phenylpropanoyl]amino]pentanedioic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3S)-3-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-4-[[(2S,3S)-1-[[(1S)-1-carboxypropyl]amino]-3-methyl-1-oxopentan-2-yl]amino]-4-oxobutanoic acid |
NA |
1262000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-4-amino-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-4-oxobutanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
711000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[4-[(2,5-dihydroxybenzoyl)amino]butanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
3013000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
273000 |
NA |
NA |
NA |
NA |
TTD |