| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
(2S)-2-[[(2S,3S)-2-[3-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]propanoylamino]-3-methylpentanoyl]amino]butanoic acid |
NA |
821000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2R)-2-[(2,5-dihydroxybenzoyl)amino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2776000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2R)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
507000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]butanoic acid |
NA |
183000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(4S)-5-[(2S)-2-[[(2S,3S)-1-[[(1S)-1-carboxypropyl]amino]-3-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-[(2,5-dihydroxybenzoyl)amino]-5-oxopentanoic acid |
NA |
3326000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
1713000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoyl]amino]butanoic acid |
NA |
137000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-5-amino-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
298000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylbutanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
318000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
422000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[6-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]hexanoylamino]butanoic acid |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3S)-3-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-4-[[(1S)-1-carboxypropyl]amino]-4-oxobutanoic acid |
NA |
680000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-(1H-imidazol-5-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2803000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[2-[(2,5-dihydroxybenzoyl)amino]acetyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2989000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2R)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]propanoyl]amino]butanoic acid |
NA |
593000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-4-amino-2-[(2,5-dihydroxybenzoyl)amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
3386000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Amino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2R)-2-(benzylcarbamoylamino)-5-(diaminomethylideneamino)-N-[2-[[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-2-oxoethyl]pentanamide |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[(2,5-dihydroxybenzoyl)amino]-3-phenylpropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
2206000 |
NA |
NA |
NA |
NA |
TTD |