| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
Tert-butyl 4-[4-[(4-carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoate;2,2,2-trifluoroacetic acid |
103000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Tert-butyl 3-[4-[(4-carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoate;2,2,2-trifluoroacetic acid |
115000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[[2-[(4-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[[2-[(4-Carbamimidoylphenyl)sulfonylamino]acetyl]amino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[3-[(4-Carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[3-[(4-Carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[4-[(4-Carbamimidoylphenyl)sulfonylamino]butanoylamino]benzoic acid;2,2,2-trifluoroacetic acid |
201000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[(4-carbamimidoylphenyl)methyl]-2-[(4-carbamimidoylphenyl)sulfonylamino]acetamide;2,2,2-trifluoroacetic acid |
125000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[3-[2-[(4-methylphenyl)methyl]-3,9-dioxo-1H-chromeno[2,3-c]pyrrol-1-yl]phenyl] hydrogen sulfate |
NA |
743000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[4-[[3-[1,3-Dioxo-5-[(4-sulfooxyphenyl)carbamoyl]isoindol-2-yl]benzoyl]amino]phenyl] hydrogen sulfate |
NA |
286000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[(2-aminoacetyl)amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]acetic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-6-amino-2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[[(2S)-2-amino-3-hydroxypropanoyl]amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]hexanoic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Epicatechin |
NA |
NA|150000 |
5190000|NA |
NA |
NA |
NA |
PubChem|TTD |
| F2 |
2-[[(2S,3S)-2-[[(2S)-1-[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
1141000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
257000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
672000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]amino]butanoic acid |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2R)-2-[[(2S,3S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]-3-methylpentanoyl]amino]-4-methylpentanoyl]amino]butanoic acid |
NA |
507000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{(S)-1-[1-(1-Formyl-4-guanidino-butylcarbamoyl)-1-methyl-ethylcarbamoyl]-4-guanidino-butyl}-carbamic acid tert-butyl ester |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-6-amino-2-[(2,5-dihydroxybenzoyl)amino]hexanoyl]amino]propanoyl]amino]-3-methylpentanoyl]amino]butanoic acid |
NA |
126000 |
NA |
NA |
NA |
NA |
TTD |