| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
2-[(2E)-2-carbamimidoylimino-6-hydroxy-1,3-benzothiazol-3-yl]-N-ethylacetamide |
2731000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[(4-carbamimidoylphenyl)sulfonylamino]-N-(3,4-dimethoxyphenyl)acetamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(4-carbamimidoylphenyl)sulfonylamino]-N-[(3,4-dimethoxyphenyl)methyl]propanamide |
175000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-(Phenylsulfamoyl)benzenecarboximidamide |
160000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(4-carbamimidoylphenyl)sulfonylamino]-N-(3,4-dimethoxyphenyl)propanamide |
187000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(4-Methoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(3-Methoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
223000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(4-carbamimidoylphenyl)sulfonylamino]-N-[(3,4-dimethoxyphenyl)methyl]butanamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(3-Methoxyphenyl)sulfamoyl]benzenecarboximidamide |
165000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(3,4-Dimethoxyphenyl)sulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(4-Methoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
245000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(3-Methoxyphenyl)sulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(3,4-Dimethoxyphenyl)sulfamoyl]benzenecarboximidamide |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(3-Methoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
165000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-[(3,4-Dimethoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[(4-carbamimidoylphenyl)sulfonylamino]-N-[(3,4-dimethoxyphenyl)methyl]acetamide |
172000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(4-carbamimidoylphenyl)sulfonylamino]-N-(3,4-dimethoxyphenyl)butanamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(4-Methoxyphenyl)sulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-[(3,4-Dimethoxyphenyl)methylsulfamoyl]benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Tert-butyl 4-[3-[(4-carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoate;2,2,2-trifluoroacetic acid |
174000 |
NA |
NA |
NA |
NA |
NA |
TTD |