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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F2 Sodium;(6-ethoxy-3-ethoxycarbonyl-2-methyl-1-benzofuran-5-yl) sulfate NA 19952623.15 NA NA NA NA TTD
F2 Sodium;(3-ethoxycarbonyl-2-methyl-6-propan-2-yloxy-1-benzofuran-5-yl) sulfate NA 12589254.12 NA NA NA NA TTD
F2 Sodium;[3-ethoxycarbonyl-6-(methoxymethoxy)-2-methyl-1-benzofuran-5-yl] sulfate NA 16000000 NA NA NA NA TTD
F2 Sodium;[3-ethoxycarbonyl-2-methyl-6-(morpholine-4-carbonyloxy)-1-benzofuran-5-yl] sulfate NA 25000000 NA NA NA NA TTD
F2 Sodium;[3-ethoxycarbonyl-6-(4-methoxybenzoyl)oxy-2-methyl-1-benzofuran-5-yl] sulfate NA 501187.23 NA NA NA NA TTD
F2 Sodium;(6-methoxy-2-methyl-3-prop-2-enoxycarbonyl-1-benzofuran-5-yl) sulfate NA 3000000 NA NA NA NA TTD
F2 Sodium;[6-methoxy-2-methyl-3-(morpholine-4-carbonyl)-1-benzofuran-5-yl] sulfate NA 2000000 NA NA NA NA TTD
F2 Sodium;[6-methoxy-3-(2-methoxyethoxycarbonyl)-2-[[6-methoxy-3-(2-methoxyethoxycarbonyl)-2-methyl-1-benzofuran-5-yl]oxymethyl]-1-benzofuran-5-yl] sulfate NA 375000 NA NA NA NA TTD
F2 Sodium;[6-ethoxy-3-ethoxycarbonyl-2-[(6-ethoxy-3-ethoxycarbonyl-2-methyl-1-benzofuran-5-yl)oxymethyl]-1-benzofuran-5-yl] sulfate NA 121000 NA NA NA NA TTD
F2 Sodium;[3-ethoxycarbonyl-6-methoxy-2-(morpholin-4-ylmethyl)-1-benzofuran-5-yl] sulfate NA 7000000 NA NA NA NA TTD
F2 Sodium;[3-ethoxycarbonyl-2-[[3-ethoxycarbonyl-6-methoxy-2-(morpholin-4-ylmethyl)-1-benzofuran-5-yl]oxymethyl]-6-methoxy-1-benzofuran-5-yl] sulfate NA 129000 NA NA NA NA TTD
F2 Sodium;[6-methoxy-2-[[6-methoxy-2-methyl-3-(morpholine-4-carbonyl)-1-benzofuran-5-yl]oxymethyl]-3-(morpholine-4-carbonyl)-1-benzofuran-5-yl] sulfate NA 7100000 NA NA NA NA TTD
F2 Sodium;[3-carboxy-2-[(3-carboxy-6-methoxy-2-methyl-1-benzofuran-5-yl)oxymethyl]-6-methoxy-1-benzofuran-5-yl] sulfate NA 371535.23 NA NA NA NA TTD
F2 Boc-Darg-Gly-Arg-Cho NA 180000 NA NA NA NA TTD
F2 ((S)-5-Amino-1-{[(1-formyl-4-guanidino-butylcarbamoyl)-methyl]-carbamoyl}-pentyl)-carbamic acid tert-butyl ester NA 400000 NA NA NA NA TTD
F2 N-[(4-carbamimidoylphenyl)methyl]-2-[(2R)-3-oxo-4-(phenacylamino)morpholin-2-yl]acetamide NA 133000 NA NA NA NA TTD
F2 4-amino-N-[(2R)-2-[2-[(4-carbamimidoylphenyl)methylamino]-2-oxoethyl]-3-oxomorpholin-4-yl]benzamide NA 150000 NA NA NA NA TTD
F2 Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD
F2 Ac-Tyr-Thr-hArg-Bn NA 1340000 NA NA NA NA TTD
F2 BnSO2-Phe-Leu-hArg-Bn NA 580000 NA NA NA NA TTD