| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
Palladium;2,10,18,26-tetrazapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(32),2,4,6,8,10,12,14,16,18,20,22,24,26,28,30-hexadecaene |
170000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Ethoxy-benzamidine |
1584893.19 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Methoxy-benzamidine |
794328.23 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[(3aS,6S,6aR)-4-[(2R,3S)-2,3-dimethylcyclopropanecarbonyl]-6-methyl-5-oxo-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrole-1-carbonyl]-N-(4-isopropylphenyl)pyrrolidine-1-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-2-[(3aS,6S,6aR)-4-(1,3-benzothiazol-2-yl)-6-methyl-5-oxo-3,3a,6,6a-tetrahydro-2H-pyrrolo[3,2-b]pyrrole-1-carbonyl]-N-(4-isopropylphenyl)pyrrolidine-1-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
5-Chlorothiophene-2-carboxamide |
431000|NA |
NA |
NA|475000|507000 |
NA |
NA |
NA |
ChEMBL|TTD |
| F2 |
3,4-Dimethylbenzene-1-carboximidamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2E)-2-cyano-3-(4-hydroxyphenyl)prop-2-enamide |
102000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2R)-2-amino-N-[3,5-bis[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]-5-(diaminomethylideneamino)pentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{[4-(N''-carbamimidoylhydrazinecarbonyl)phenyl]formohydrazido}methanimidamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-4-guanidinobutanamide |
800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-5-guanidinopentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-6-guanidinohexanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
amino-N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)butanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;[3-ethoxycarbonyl-6-[(3-ethoxycarbonyl-6-methoxy-5-sulfonatooxy-1-benzofuran-2-yl)methoxy]-2-methyl-1-benzofuran-5-yl] sulfate |
NA |
758577.58 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Disodium;[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-6-methoxy-2-methyl-1-benzofuran-5-yl)oxymethyl]-5-sulfonatooxy-1-benzofuran-6-yl] sulfate |
NA |
363078.05 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;(3-ethoxycarbonyl-6-methoxy-2-methyl-1-benzofuran-5-yl) sulfate |
NA |
2500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;(6-methoxy-3-methoxycarbonyl-2-methyl-1-benzofuran-5-yl) sulfate |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[6-methoxy-2-methyl-3-[(2-methylpropan-2-yl)oxycarbonyl]-1-benzofuran-5-yl] sulfate |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[6-methoxy-3-(2-methoxyethoxycarbonyl)-2-methyl-1-benzofuran-5-yl] sulfate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |