| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
Sodium;[6-methoxy-2-methyl-3-(piperidine-1-carbonyl)-1-benzofuran-5-yl] sulfate |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
H-Phe-Phe-hArg-Bn |
NA |
1480000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
BnSO2-Phe-Phe-hArg-Bn |
NA |
590000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
H-Tyr-Thr-hArg-Bn |
NA |
1340000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Ac-Phe-Phe-hArg-Bn |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Cbz-D-Phe-Phe-hArg-Bn |
NA |
560000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
BnSO2-D-Phe-Phe-hArg-Bn |
NA |
640000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Cbz-Phe-Phe-hArg-Bn |
NA |
650000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-(Benzylsulfamoyl)benzenecarboximidamide |
230000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-(Phenylsulfamoyl)benzenecarboximidamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Methyl 3-[4-[(6-carbamoylnaphthalene-2-carbonyl)amino]phenyl]benzoate |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
6-amino-N-[(3S,7E,9S,12R,16S,19S)-16-[[3-(aminomethyl)phenyl]methyl]-12-[(2S)-butan-2-yl]-9-[(4-hydroxyphenyl)methyl]-2,6,11,14,18-pentaoxo-1,5,10,13,17-pentazabicyclo[17.3.0]docos-7-en-3-yl]hexanamide |
330000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[(2R)-1-[4-(2-hydroxyethyl)piperidin-1-yl]-1-oxo-3-pyridin-4-ylpropan-2-yl]-3,3-dimethyl-2,4-dihydro-1H-quinoline-8-sulfonamide |
132700 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[(3S,7E,9S,12R,16S,19S)-16-[[3-(aminomethyl)phenyl]methyl]-12-[(2S)-butan-2-yl]-9-[(4-hydroxyphenyl)methyl]-2,6,11,14,18-pentaoxo-1,5,10,13,17-pentazabicyclo[17.3.0]docos-7-en-3-yl]acetamide |
680000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-Cyano-3-(4-isopropylphenyl)-N-(tetrahydro-2-furanylmethyl)acrylamide |
165000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-Methyl-benzamidine |
100000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3S,3aR,6aS)-1-Cyclopropanecarbonyl-4-[(S)-1-(5-dimethylamino-naphthalene-1-sulfonyl)-pyrrolidine-2-carbonyl]-3-methyl-hexahydro-pyrrolo[3,2-b]pyrrol-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(3R)-2-[2-(4-chlorophenyl)acetyl]-N-[4-(3-oxomorpholin-4-yl)phenyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-(7-Carbamimidoyl-naphthalen-2-yl)-2-{4-[(S)-1-(1-imino-ethyl)-pyrrolidin-3-yloxy]-phenyl}-propionic acid |
NA |
1200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
ethyl 2-[(2E)-2-carbamimidoylimino-6-hydroxy-1,3-benzothiazol-3-yl]acetate |
481000 |
NA |
NA |
NA |
NA |
NA |
TTD |