| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
N-[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-methyl]-carbamoyl}-3-(1-oxy-pyridin-2-yl)-propyl]-malonamic acid |
140000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
[1-{[(2-Aminomethyl-5-chloro-benzylcarbamoyl)-methyl]-carbamoyl}-3-(1-oxy-pyridin-2-yl)-propylamino]-acetic acid |
125000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(4-Guanidino-benzyl)-carbamic acid benzyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-2-[(3R)-3-[3-(diaminomethylideneamino)propyl]-2-oxopiperazin-1-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-(2-phenoxyethyl)pyridin-4-amine |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-(Naphthalene-2-sulfonylamino)-N-[(S)-1-(piperidine-1-carbonyl)-3-(pyridin-4-ylamino)-propyl]-acetamide |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Amino-N-{3-[(S)-2-[4-(2-amino-ethyl)-piperidin-1-yl]-1-(3-aminomethyl-benzyl)-2-oxo-ethylsulfamoyl]-phenyl}-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Amino-N-{3-[(S)-2-[4-(2-amino-ethyl)-piperidin-1-yl]-1-(4-aminomethyl-benzyl)-2-oxo-ethylsulfamoyl]-phenyl}-propionamide |
325000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-1-[(2S)-2-[[3-(3-aminopropanoylamino)phenyl]sulfonylamino]-3-(3-carbamimidoylphenyl)propanoyl]piperidine-2-carboxylic acid |
159000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-(Hydroxymethyl)Benzamidine |
3162277.66 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-N-(3-chlorobenzyl)-1-acetylpyrrolidine-2-carboxamide |
1460000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-N-(3-chlorobenzyl)-1-propionylpyrrolidine-2-carboxamide |
330000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-1-butyryl-N-(3-chlorobenzyl)pyrrolidine-2-carboxamide |
322000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-N-(3-chlorobenzyl)-1-(3-methylbutanoyl)pyrrolidine-2-carboxamide |
155000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-N-(3-chlorobenzyl)-1-(3,3-dimethylbutanoyl)pyrrolidine-2-carboxamide |
484000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(R)-2-(3-acetamido-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)-N-((6-amino-2-methylpyridin-3-yl)methyl)acetamide, trifluoroacetate |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-2-(3-acetamido-4-oxo-3,4-dihydrobenzo[b][1,4]thiazepin-5(2H)-yl)-N-((6-amino-2-methylpyridin-3-yl)methyl)acetamide, trifluoroacetate |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(R)-4-(5-(2-(4-carbamimidoylbenzylamino)-2-oxoethyl)-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]thiazepin-3-ylamino)-4-oxobutanoic acid, trifluoroacetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(S)-5-guanidino-N-((S)-1-((S)-5-guanidino-1-(3-guanidinopropylamino)-1-oxopentan-2-ylamino)-3-methyl-1-oxobutan-2-yl)-2-(2-phenylacetamido)pentanamide |
102000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-Bromo-benzamidine |
1584893.19 |
NA |
NA |
NA |
NA |
NA |
TTD |