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drugs and pathways
negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
F7
Ac-Tyr-Thr-hArg-Bn
NA
1340000
NA
NA
NA
NA
TTD
F7
BnSO2-Phe-Leu-hArg-Bn
NA
580000
NA
NA
NA
NA
TTD
F7
H-Phe-Phe-hArg-Bn
NA
1480000
NA
NA
NA
NA
TTD
F7
H-Tyr-Thr-hArg-Bn
NA
1340000
NA
NA
NA
NA
TTD
F7
Ac-Phe-Phe-hArg-Bn
NA
400000
NA
NA
NA
NA
TTD
F7
BnSO2-D-Phe-Phe-hArg-Bn
NA
640000
NA
NA
NA
NA
BindingDB|TTD
F7
Cbz-Phe-Phe-hArg-Bn
NA
109000
NA
NA
NA
NA
BindingDB
F7
(3R)-2-[2-(4-chlorophenyl)acetyl]-N-[4-(3-oxomorpholin-4-yl)phenyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide
NA
1000000
NA
NA
NA
NA
TTD
F7
5-Chlorobenzotriazole
8700000
NA
NA
NA
NA
NA
BindingDB
F7
Ethyl {(1S)-5-amino-1-[(5-{4-[(2,3-dihydro-1H-inden-2-ylamino)carbonyl]benzyl}-1,2,4-oxadiazol-3-YL)carbonyl]pentyl}carbamate
150000
NA
NA
NA
NA
NA
TTD
F7
N-[3-[(4-fluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide
250000
NA
NA
NA
NA
NA
TTD
F7
N-[3-[(3-fluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide
250000
NA
NA
NA
NA
NA
TTD
F7
N-[3-[(2-fluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide
250000
NA
NA
NA
NA
NA
TTD
F7
N-[3-[(3,5-difluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide
250000
NA
NA
NA
NA
NA
TTD
F7
N-[3-[(3,4-dimethoxyphenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide
250000
NA
NA
NA
NA
NA
TTD
F7
1-Aminoisoquinoline
4000000
NA
NA
NA
NA
NA
BindingDB
F7
5-Chloroindole-2-carboxylic acid
3500000
NA
NA
NA
NA
NA
BindingDB
F7
5-Chloroindole
4300000
NA
NA
NA
NA
NA
BindingDB
F7
Niacinamide
8000000
NA
NA
NA
NA
NA
BindingDB|PubChem
F7
1-(1-Naphthyl)ethanol
16000000
NA
NA
NA
NA
NA
BindingDB
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