| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FAAH |
N-[2-[bis(4-phenylmethoxyphenyl)methyl-methylamino]ethyl]-4-cyano-N-methylpyrazole-1-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FAAH |
N-[2-[bis(4-phenylmethoxyphenyl)methyl-methylamino]ethyl]-N,4-dimethylpyrazole-1-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FAAH |
N-[2-[bis(4-phenylmethoxyphenyl)methyl-methylamino]ethyl]-N-methylpyrazole-1-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FAAH |
Disulfiram |
NA |
363078 |
NA |
NA |
NA |
NA |
PubChem |
| FAAH |
Ibuprofen Sodium |
NA |
380189 |
NA |
NA |
NA |
NA |
PubChem |
| FAAH |
Dipentamethylenethiuram disulfide |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FAAH |
Bis(dimethylthiocarbamoyl) sulfide |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FABP1 |
Tacrine |
NA |
NA |
900000|9e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL|PubChem |
| FABP1 |
2-Benzylaminopyridine |
NA |
NA |
300000|3e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FABP1 |
[4-(1,3-Benzodioxol-5-ylmethyl)piperazin-1-yl](furan-2-yl)methanone |
NA |
NA |
400000|4e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FABP3 |
Fabp4/5-IN-5 |
NA |
103700 |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
5-[[4-(3-Chloro-4-fluorophenyl)naphthalen-1-yl]sulfonylamino]-2-fluorobenzoic acid |
NA |
103050 |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
(2S,4S)-3-[(2-cyano-5-phenylphenyl)carbamoyl]-2,4-diphenylcyclobutane-1-carboxylic acid |
127000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
(2R,4R)-3-[[2-cyano-5-(3,6-dihydro-2H-pyran-4-yl)phenyl]carbamoyl]-2,4-diphenylcyclobutane-1-carboxylic acid |
116200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
(2R,4R)-3-[[3-(2-oxo-1,3-dihydroindol-6-yl)phenyl]carbamoyl]-2,4-diphenylcyclobutane-1-carboxylic acid |
291600 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
Elaidate |
NA |
NA |
359000 |
NA |
NA |
NA |
BindingDB |
| FABP3 |
5-[2-[5-(4-Chlorophenyl)-1-phenylpyrazol-3-yl]phenoxy]pentanoic acid |
NA |
243000 |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
4-[2-[5-(4-Methylphenyl)-1-phenylpyrazol-3-yl]phenoxy]butanoic acid |
NA |
4730000 |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
4-[2-[5-(4-Bromophenyl)-1-phenylpyrazol-3-yl]phenoxy]butanoic acid |
NA |
224000 |
NA |
NA |
NA |
NA |
BindingDB |
| FABP3 |
4-[2-[1-(2-Methoxyphenyl)-5-phenylpyrazol-3-yl]phenoxy]butanoic acid |
NA |
505000 |
NA |
NA |
NA |
NA |
BindingDB |