| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FABP4 |
2-[2-[5-(4-Chlorophenyl)-1-phenylpyrazol-3-yl]phenoxy]acetic acid |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| FABP4 |
5-[2-[5-(4-Methylphenyl)-1-phenylpyrazol-3-yl]phenoxy]pentanoic acid |
NA |
259000 |
NA |
NA |
NA |
NA |
TTD |
| FABP6 |
N-benzyl-1-methylsulfonylazepan-4-amine |
NA |
NA |
3e+05 |
NA |
NA |
NA |
ChEMBL |
| FABP6 |
4-[(5,6-Dimethylbenzimidazol-1-yl)methyl]-2-methyl-1,3-thiazole |
NA |
NA |
4e+05 |
NA |
NA |
NA |
ChEMBL |
| FABP6 |
Tacrine |
NA |
NA |
2e+05|200000 |
NA |
NA |
NA |
ChEMBL|PubChem |
| FABP6 |
2-Benzylaminopyridine |
NA |
NA |
3e+05 |
NA |
NA |
NA |
ChEMBL |
| FABP6 |
1-(4-chlorobenzyl)-5-[(4-methylpiperazino)carbonyl]-2(1H)-pyridinone |
NA |
NA |
210000 |
NA |
NA |
NA |
ChEMBL |
| FABP6 |
[4-(2-Methylbenzyl)piperazin-1-yl](pyridin-3-yl)methanone |
NA |
NA |
290000 |
NA |
NA |
NA |
ChEMBL |
| FABP6 |
[4-(1,3-Benzodioxol-5-ylmethyl)piperazin-1-yl](furan-2-yl)methanone |
NA |
NA |
210000 |
NA |
NA |
NA |
ChEMBL |
| FABP7 |
(2S,4S)-3-[(2-cyano-5-phenylphenyl)carbamoyl]-2,4-diphenylcyclobutane-1-carboxylic acid |
101590 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FADS1 |
Mk-8245 |
NA |
100000000 |
NA |
NA |
NA |
NA |
PubChem |
| FADS2 |
1-[5-(2H-Tetrazol-5-yl)-1,3,4-thiadiazol-2-yl}-4-[2-(trifluoromethyl)phenoxy]piperidine |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| FADS2 |
2-Methyl-5-(6-(4-(2-(trifluoromethyl)phenoxy)piperidin-1-yl)pyridazin-3-yl)-1,3,4-thiadiazole |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| FADS2 |
2-(5-(5-(4-(2-Bromo-5-fluorophenoxy)piperidin-1-yl)-1,3,4-thiadiazol-2-yl)-2H-tetrazol-2-yl)acetic acid |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| FADS2 |
Mk-8245 |
NA |
100000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FADS2 |
4-(2-Bromo-5-fluorophenoxy)-1-[5-(2H-tetrazol-5-yl)-1,3,4-thiadiazol-2-yl]piperidine |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| FAP |
2-Pyrrolidinecarbonitrile, 1-((2S)-2-amino-3,3-dimethyl-1-oxobutyl)-, (2S)- |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
Saxagliptin |
NA |
1720000 |
NA |
NA |
NA |
NA |
PubChem |
| FAP |
Alogliptin |
NA |
1470000 |
NA |
NA |
NA |
NA |
PubChem |
| FAP |
(2S,3aS,6aS)-1-[(3R)-3-amino-4-(2-methylphenyl)butanoyl]-3,3a,4,5,6,6a-hexahydro-2H-cyclopenta[b]pyrrole-2-carbonitrile |
NA |
109880 |
NA |
NA |
NA |
NA |
BindingDB|TTD |