| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FASN |
(2R,3R,4S,5S)-2-(6-aminopurin-9-yl)-5-(methylsulfonylmethyl)oxolane-3,4-diol |
220000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FASN |
[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-dimethylsulfanium;iodide |
2500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FASN |
Methionine |
150000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FAU |
NB-124 sulfate |
NA |
1493000 |
NA |
NA |
NA |
NA |
PubChem |
| FBP1 |
Urea, 1-propyl-3-(m-tolylsulfonyl)- |
NA |
320180 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
Disulfiram |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FBP1 |
2-(6-amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-9H-purin-8-ylamino)ethyl dihydrogen phosphate |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
{[(6-Amino-9-phenethyl-9H-purin-8-ylmethyl)-amino]-methyl}-phosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[2-(6-Amino-9-phenethyl-9H-purin-8-ylsulfanyl)-ethyl]-phosphonic Acid |
NA |
145000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
5-(6-Amino-9-phenethyl-9H-purin-8-yl)-furan-2-sulfonic Acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[5-(6-Dimethylamino-9-phenethyl-9H-purin-8-yl)-furan-2-yl]-phosphonic Acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[2-(6-Amino-9-phenethyl-9H-purine-8-sulfonyl)-ethyl]-phosphonic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
1-(3-Chlorophenylsulfonyl)-3-propylurea |
NA |
234231 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
1-Butyl-3-(3-chlorophenylsulfonyl)urea |
NA |
134180 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
1-(3-Chlorophenylsulfonyl)-3-(2-(methylthio)ethyl)urea |
NA |
277143 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[3-(6-Amino-9-phenethyl-9H-purin-8-yl)-propyl]-phosphinic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[2-(6-Amino-9-phenethyl-9H-purin-8-yl)-1-methyl-ethyl]-phosphinic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
[2-(6-Amino-9-phenethyl-9H-purin-8-yl)-ethoxy]-phosphinic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-9-yl dihydrogen phosphate |
NA |
335000 |
NA |
NA |
NA |
NA |
TTD |
| FBP1 |
2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-7-ylphosphonic acid |
NA |
354000 |
NA |
NA |
NA |
NA |
TTD |