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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
FBP1 2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-9-ylphosphonic acid NA 354000 NA NA NA NA TTD
FBP1 2-amino-8H-indeno[1,2-d]thiazol-6-yl dihydrogen phosphate NA 146000 NA NA NA NA TTD
FBP1 2-amino-8H-indeno[1,2-d]thiazol-5-yl dihydrogen phosphate NA 307000 NA NA NA NA TTD
FBP1 2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-7-yl dihydrogen phosphate NA 112000 NA NA NA NA TTD
FBP1 (2-amino-8H-indeno[1,2-d]thiazol-6-yloxy)methylphosphonic acid NA 112000 NA NA NA NA TTD
FBP1 (2-amino-8H-indeno[1,2-d]thiazol-5-yloxy)methylphosphonic acid NA 112000 NA NA NA NA TTD
FBP2 Urea, 1-propyl-3-(m-tolylsulfonyl)- NA 320180 NA NA NA NA TTD
FBP2 2-(6-amino-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-9H-purin-8-ylamino)ethyl dihydrogen phosphate NA 140000 NA NA NA NA TTD
FBP2 {[(6-Amino-9-phenethyl-9H-purin-8-ylmethyl)-amino]-methyl}-phosphonic acid NA 500000 NA NA NA NA TTD
FBP2 [2-(6-Amino-9-phenethyl-9H-purin-8-ylsulfanyl)-ethyl]-phosphonic Acid NA 145000 NA NA NA NA TTD
FBP2 5-(6-Amino-9-phenethyl-9H-purin-8-yl)-furan-2-sulfonic Acid NA 150000 NA NA NA NA TTD
FBP2 [5-(6-Dimethylamino-9-phenethyl-9H-purin-8-yl)-furan-2-yl]-phosphonic Acid NA 250000 NA NA NA NA TTD
FBP2 [2-(6-Amino-9-phenethyl-9H-purine-8-sulfonyl)-ethyl]-phosphonic Acid NA 1000000 NA NA NA NA TTD
FBP2 1-(3-Chlorophenylsulfonyl)-3-propylurea NA 234231 NA NA NA NA TTD
FBP2 1-Butyl-3-(3-chlorophenylsulfonyl)urea NA 134180 NA NA NA NA TTD
FBP2 1-(3-Chlorophenylsulfonyl)-3-(2-(methylthio)ethyl)urea NA 277143 NA NA NA NA TTD
FBP2 [3-(6-Amino-9-phenethyl-9H-purin-8-yl)-propyl]-phosphinic Acid NA 1000000 NA NA NA NA TTD
FBP2 [2-(6-Amino-9-phenethyl-9H-purin-8-yl)-1-methyl-ethyl]-phosphinic Acid NA 1000000 NA NA NA NA TTD
FBP2 [2-(6-Amino-9-phenethyl-9H-purin-8-yl)-ethoxy]-phosphinic Acid NA 1000000 NA NA NA NA TTD
FBP2 2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-9-yl dihydrogen phosphate NA 335000 NA NA NA NA TTD