| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FAP |
(2S,3aS,6aS)-1-[(3R)-3-amino-4-(4-fluorophenyl)butanoyl]-3,3a,4,5,6,6a-hexahydro-2H-cyclopenta[b]pyrrole-2-carbonitrile |
NA |
153700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FAP |
[4-[[(2S)-5-(carbamoylamino)-2-[[(2S)-2-[6-(2,5-dioxopyrrol-1-yl)hexanoylamino]-3-methylbutanoyl]amino]pentanoyl]amino]phenyl]methyl (2R)-2-[[(3S)-1-[[(1R,3R)-1-[4-[[(2R,4S)-1-(4-hydroxyphenyl)-5-methoxy-4-methyl-5-oxopentan-2-yl]carbamoyl]-1,3-thiazol-2-yl]-4-methyl-1-propoxypentan-3-yl]-propylamino]-3-methyl-1-oxopentan-2-yl]carbamoyl]piperidine-1-carboxylate |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 5349 |
NA |
14000000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 4949 |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 4367 |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 5552 |
NA |
41070000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 1049 D |
NA |
640000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 4160 |
NA |
2200000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
US11096924, DASH-inhibitors 4312 |
NA |
13000000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
Leu-boroPro |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
1G244 |
NA |
2200000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
Ala-boroPro thioxoamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| FAP |
Glu-boroSar |
NA |
11000000 |
NA |
NA |
NA |
NA |
BindingDB |
| FASN |
L-Methionine methylsulfonium iodide |
140000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FASN |
Methylthioadenosine sulfoxide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FASN |
(+)-Epicatechin |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FASN |
Orlistat |
NA |
203000 |
NA |
NA |
NA |
NA |
PubChem |
| FASN |
Lansoprazole |
NA |
124000 |
NA |
NA |
NA |
NA |
PubChem |
| FASN |
S-Adenosylhomocysteine |
150000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FASN |
5'-Methylthioadenosine |
1500000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |