| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FBP2 |
2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-7-ylphosphonic acid |
NA |
354000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-9-ylphosphonic acid |
NA |
354000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
2-amino-8H-indeno[1,2-d]thiazol-6-yl dihydrogen phosphate |
NA |
146000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
2-amino-8H-indeno[1,2-d]thiazol-5-yl dihydrogen phosphate |
NA |
307000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
2-Amino-4,5-dihydronaphtho[1,2-d]thiazol-7-yl dihydrogen phosphate |
NA |
112000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
(2-amino-8H-indeno[1,2-d]thiazol-6-yloxy)methylphosphonic acid |
NA |
112000 |
NA |
NA |
NA |
NA |
TTD |
| FBP2 |
(2-amino-8H-indeno[1,2-d]thiazol-5-yloxy)methylphosphonic acid |
NA |
112000 |
NA |
NA |
NA |
NA |
TTD |
| FCER1A |
Ikcnckrhvikphicrkicgan-NH2 |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB |
| FCER1A |
Ikcnckrhvikphicrkicgkn-NH2 |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB |
| FCER1A |
Ikcnckrhviaphicrkicgkn-NH2 |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB |
| FCER1A |
Ikcnckrhvikphicraicgkn-NH2 |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB |
| FCGRT |
Ctghfgglypcngp |
NA |
239000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FCGRT |
Ctghfgglypc |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FCGRT |
Tghfgglyp |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FCGRT |
H-Arg-Phe-Pen-Thr-Gly-N(Me)His-Phe-Gly-Gly-Leu-Tyr-Pro-Cys-OH |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FCGRT |
H-Gln-Arg-Phe-Pen-Thr-Gly-His-Phe-Gly-Gly-Leu-Phe(4-NO2)-Pro-Cys-Asn-Gly-Pro-OH |
NA |
NA|122000 |
180000|NA |
NA |
NA |
NA |
BindingDB|TTD |
| FCGRT |
(2S)-1-[2-[[(2S)-4-amino-2-[[(2R)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2R)-2-[[(2S)-2-[[(2S)-5-carbamimidamido-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]amino]-3-phenylpropanoyl]amino]-3-methyl-3-sulfanylbutanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxy-2-nitrophenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-sulfanylpropanoyl]amino]-4-oxobutanoyl]amino]acetyl]pyrrolidine-2-carboxylic acid |
NA |
NA|125000 |
290000|NA |
NA |
NA |
NA |
BindingDB|TTD |
| FCGRT |
H-Arg-Phe-Pen-Thr-Gly-Ala(pyrrol-3-yl)(pyrrol-3-yl)-Phe-Gly-Sar-N(Me)Leu-Tyr-Pro-Cys-OH |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FCGRT |
(2R)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[4-[[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-3-phenylpropanoyl]amino]-3-methyl-3-sulfanylbutanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]methyl]benzoyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-sulfanylpropanoic acid |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| FCGRT |
(2R)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[4-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2R)-2-[[(2S)-2-[[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-3-phenylpropanoyl]amino]-3-methyl-3-sulfanylbutanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]phenyl]acetyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-sulfanylpropanoic acid |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |