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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
FCGRT (2S)-1-[2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2S)-3-amino-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]amino]-3-phenylpropanoyl]amino]propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]-4-oxobutanoyl]amino]acetyl]pyrrolidine-2-carboxylic acid NA 120000 NA NA NA NA BindingDB
FCGRT (2S)-1-[2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]amino]-3-phenylpropanoyl]amino]pentanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-carboxypropanoyl]amino]-4-oxobutanoyl]amino]acetyl]pyrrolidine-2-carboxylic acid NA 120000 NA NA NA NA BindingDB
FCGRT (2S)-1-[2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2,5-diamino-5-oxopentanoyl]amino]pentanoyl]amino]-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-4-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxypropanoyl]amino]-4-oxobutanoyl]amino]acetyl]pyrrolidine-2-carboxylic acid NA NA 230000 NA NA NA BindingDB
FDPS 2-Hydroxy-2-phosphono-3-(pyridin-3-yl)propanoic acid NA 200000|253500|254000|467000 NA NA NA NA BindingDB
FDPS [Aminomethyl(hydroxy)phosphoryl]methylphosphonic acid NA 150000 NA NA NA NA BindingDB
FDPS Pyrophosphoric acid NA 243000|181000 NA NA NA NA PubChem
FDPS N(6)-Isopentenyladenosine NA NA 550000|1210000|2020000|2210000 NA NA NA BindingDB
FDPS 2-Hydroxy-3-(1-oxidopyridin-1-ium-3-yl)-2-phosphonopropanoic acid NA 2000000 NA NA NA NA BindingDB|TTD
FDPS 3-(1-Oxidopyridin-1-ium-3-yl)-2-phosphonopropanoic acid NA 2000000 NA NA NA NA TTD
FDPS [[Hydroxy(methyl)phosphoryl]-[(3-methylpyridin-2-yl)amino]methyl]-methylphosphinic acid NA 330000 NA NA NA NA BindingDB
FDPS [Acetamidomethyl(hydroxy)phosphoryl]methylphosphonic acid NA 177000 NA NA NA NA BindingDB
FDPS [(Diaminomethylideneamino)methyl-hydroxyphosphoryl]methylphosphonic acid NA 233000 NA NA NA NA BindingDB
FDPS 2-Phosphono-3-pyridin-3-ylpropanoic acid NA 1000000 NA NA NA NA BindingDB|TTD
FDPS 2-(5-Chloro-1-benzothiophen-3-yl)acetic acid NA 500000000 NA NA NA NA TTD
FDPS 2,5-bis[[4-(4,5-dihydro-1H-imidazol-2-yl)phenyl]carbamoyl]-N-hydroxybenzeneamine oxide NA 109000 NA NA NA NA BindingDB
FDPS 2-Chloro-3-(3-pyridinyl)-2-phosphonopropionic acid NA 600000 NA NA NA NA TTD
FDPS 2-Fluoro-3-(3-pyridinyl)-2-phosphonopropionic acid NA 600000 NA NA NA NA TTD
FDPS Riboprine NA NA 550000|2210000|2020000|1210000 NA NA NA PubChem
FDPS {2-[3-(Decyloxy)phenyl]-1-hydroxy-1-phosphonoethyl}phosphonic acid NA 550000 NA NA NA NA BindingDB|TTD
FDPS [Hydroxy(oxido)phosphoryl] phosphate NA 181000|243000 NA NA NA NA BindingDB