| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FDPS |
P,P'-(1-Aminopropylidene)bis(phosphonic acid) |
NA |
149590 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FDPS |
(1-Phosphono-butyl)-phosphonic acid |
NA |
150360 |
NA |
NA |
NA |
NA |
BindingDB |
| FDPS |
2-Pyridin-3-ylethylphosphonic acid |
NA|128300 |
824000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FDPS |
Tianafac |
NA |
500000000 |
NA |
NA |
NA |
NA |
TTD |
| FDPS |
(2S)-1-[(benzyloxy)carbonyl]-2,3-dihydro-1H-indole-2-carboxylic acid |
NA |
500000000 |
NA |
NA |
NA |
NA |
TTD |
| FDPS |
2-(6-Methoxy-1-benzofuran-3-yl)acetic acid |
NA |
500000000 |
NA |
NA |
NA |
NA |
TTD |
| FFAR1 |
Setogepram |
NA |
NA |
NA |
1047129 |
NA |
NA |
GtoPDB |
| FFAR1 |
Pioglitazone |
NA |
NA |
NA |
812831 |
NA |
NA |
PubChem |
| FFAR2 |
Propionic Acid |
NA |
NA|130000 |
NA |
250000|257040|NA |
NA |
NA |
BindingDB|PubChem|TTD |
| FFAR2 |
Acetic Acid |
NA |
NA|120000 |
NA |
250000|NA |
NA |
NA |
BindingDB|PubChem|TTD |
| FFAR2 |
(S)-2-(4-chlorophenyl)-4-methoxy-N-(thiazol-2-yl)butanamide |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FFAR3 |
5-cyano-2,6-dimethyl-N-(2-methylphenyl)-4-(2-methylpropyl)-1,4-dihydropyridine-3-carboxamide |
NA |
NA |
NA |
102329 |
NA |
NA |
BindingDB |
| FFAR3 |
1-Methylcyclopropanecarboxylic acid |
NA |
NA |
NA |
131826 |
NA |
NA |
BindingDB |
| FGD1 |
Cyclopentenyluracil |
230000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FGF1 |
(2R,3S,4R)-4-(3-phenoxypropoxy)-2-[(sulfonatooxy)methyl]tetrahydro-2H-pyran-3-yl sulfate |
NA |
NA |
3250000 |
NA |
NA |
NA |
BindingDB |
| FGF1 |
(2R,3S,4R)-4-(benzyloxy)-2-[(sulfonatooxy)methyl]tetrahydro-2H-pyran-3-yl sulfate |
NA |
NA |
3410000 |
NA |
NA |
NA |
BindingDB |
| FGF1 |
3-(allyloxy)-6-methoxy-2-methyl-5-(sulfonatooxy)tetrahydro-2H-pyran-4-yl sulfate |
NA |
NA |
1340000 |
NA |
NA |
NA |
BindingDB |
| FGF1 |
3-(benzyloxy)-6-methoxy-2-methyl-5-(sulfonatooxy)tetrahydro-2H-pyran-4-yl sulfate |
NA |
NA |
337500 |
NA |
NA |
NA |
BindingDB |
| FGF1 |
2-(Benzyloxy)-3-methoxy-6,8-dioxabicyclo[3.2.1]oct-4-yl sulfate |
NA |
NA |
307000 |
NA |
NA |
NA |
BindingDB |
| FGF1 |
(2R,3R,4R)-4-methoxy-2-[(sulfonatooxy)methyl]tetrahydro-2H-pyran-3-yl sulfate |
NA |
NA |
5940000 |
NA |
NA |
NA |
BindingDB |