| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FGFR1 |
Kinase inhibitor, D1 |
NA |
469000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR1 |
4-Amino-1-[[2-(2-octadecoxyethoxy)-2-oxo-1,4,2lambda5-dioxaphosphinan-5-yl]methyl]pyrimidin-2-one |
NA |
NA |
NA |
300000 |
NA |
NA |
BindingDB |
| FGFR1 |
4-Amino-1-[[2-(3-hexadecoxypropoxy)-2-oxo-1,4,2lambda5-dioxaphosphinan-5-yl]methyl]pyrimidin-2-one |
NA |
NA |
NA |
300000 |
NA |
NA |
BindingDB |
| FGFR1 |
4-Amino-1-[[2-(3-octadecoxypropoxy)-2-oxo-1,4,2lambda5-dioxaphosphinan-5-yl]methyl]pyrimidin-2-one |
NA |
NA |
NA |
300000 |
NA |
NA |
BindingDB |
| FGFR2 |
4-[3-(4-aminophenyl)-1H-indazol-6-yl]phenol |
NA |
198000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FGFR2 |
2-fluoro-4-[3-(4-piperazin-1-ylphenyl)-1H-indazol-6-yl]phenol |
NA |
258000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR3 |
Fgfr2-IN-2 |
NA |
758000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR3 |
4-[3-[4-(4-ethylpiperazin-1-yl)phenyl]-1H-indazol-6-yl]phenol |
NA |
501000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR3 |
2-fluoro-4-[3-(4-piperazin-1-ylphenyl)-1H-indazol-6-yl]phenol |
NA |
753000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR3 |
3-fluoro-4-[3-(4-piperazin-1-ylphenyl)-1H-indazol-6-yl]phenol |
NA |
915000 |
NA |
NA |
NA |
NA |
BindingDB |
| FGFR3 |
6-Quinoxalinamine |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| FGR |
Linifanib |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FIBCD1 |
Acetic Acid |
NA |
3000000 |
NA |
NA |
NA |
NA |
PubChem |
| FIBCD1 |
Acetylcholine |
NA |
10000000 |
NA |
NA |
NA |
NA |
PubChem |
| FIBCD1 |
N-Acetyl-D-Glucosamine |
NA |
4000000 |
NA |
NA |
NA |
NA |
PubChem |
| FIBCD1 |
N-Acetyl-D-Mannosamine |
NA |
2000000 |
NA |
NA |
NA |
NA |
PubChem |
| FIBCD1 |
N-Acetyl-L-alanine |
NA |
4000000 |
NA |
NA |
NA |
NA |
PubChem |
| FKBP1A |
1-Benzyl-4-[(R)-2-((1S,3S,5S)-3,5-dimethyl-2-oxo-cyclohexyl)-2-hydroxy-ethyl]-piperidine-2,6-dione |
NA |
116700 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FKBP1A |
4-[(R)-2-((1S,3S,5S)-3,5-Dimethyl-2-oxo-cyclohexyl)-2-hydroxy-ethyl]-1-methyl-piperidine-2,6-dione |
NA |
124100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FKBP1A |
Cycloheximide acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |