| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FKBP1A |
N-(3-chloro-4-methylphenyl)piperidine-1-sulfonamide |
NA |
NA |
135000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(4-Isopropyl-3-methylphenoxy)-1-morpholinoethanone |
NA |
NA |
187000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
N-cyclopentyl-4-[2-(morpholin-4-yl)-2-oxoethoxy]benzenesulfonamide |
NA |
NA |
755000 |
NA |
NA |
NA |
BindingDB |
| FKBP1A |
3-(4-Methoxyphenyl)-1-morpholin-4-ylpropan-1-one |
NA |
NA |
204000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
1-(2,6-Dimethylmorpholin-4-yl)-2-(phenylsulfanyl)ethanone |
NA |
NA |
726000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(2-Morpholino-2-oxoethylthio)-5-(trifluoromethyl)benzoic acid |
NA |
NA |
453000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(4-Chloro-3-isopropyl-5-methylphenoxy)-1-morpholinoethanone |
NA |
NA |
576000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
3-methyl-4-(2-morpholino-2-oxoethoxy)-N-(3-(trifluoromethyl)phenyl)benzenesulfonamide |
NA |
NA |
576000 |
NA |
NA |
NA |
BindingDB |
| FKBP1A |
(S)-1-[2-((1S,2R,5R)-1-Hydroxy-5-isopropyl-2-methyl-cyclohexyl)-2-oxo-acetyl]-piperidine-2-carboxylic acid benzyl ester |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FKBP1A |
1-(Morpholin-4-yl)-3-phenylpropan-1-one |
NA |
NA |
578000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
4-((R)-2-Hydroxy-2-{(1R,3S,5S)-2-[(Z)-hydroxyimino]-3,5-dimethyl-cyclohexyl}-ethyl)-piperidine-2,6-dione |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB |
| FKBP1A |
2-(Benzo[d][1,3]dioxol-5-yloxy)-1-morpholinoethanone |
NA |
NA |
576000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
N-(3,5-dichlorophenyl)piperidine-1-sulfonamide |
NA |
NA |
155000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(3-Chlorophenoxy)-1-morpholinoethanone |
NA |
NA |
755000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
4-{[(4'-Methyl-4-biphenylyl)oxy]acetyl}morpholine |
NA |
NA |
755000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
N-(4-fluorophenyl)piperidine-1-sulfonamide |
NA |
NA |
319000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
4-[(4-Ethoxyphenoxy)acetyl]morpholine |
NA |
NA |
576000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(4-Chloro-3,5-dimethylphenoxy)-1-morpholinoethanone |
NA |
NA |
231000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
2-(4-Ethylphenoxy)-1-morpholinoethanone |
NA |
NA |
123000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| FKBP1A |
Morpholine, 4-((4-methoxyphenoxy)acetyl)- |
NA |
NA |
357000 |
NA |
NA |
NA |
BindingDB|ChEMBL |