Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| GABRA4 | Temazepam | NA | 62517300 | NA | NA | NA | NA | PubChem |
| GABRA4 | Methyl(piperidin-4-yl)phosphinic acid | 340000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA4 | Piperidin-4-yl-phosphinic acid | NA | NA | NA | 140000 | NA | NA | BindingDB |
| GABRA4 | 7-Aminoflunitrazepam | NA | 15381500 | NA | NA | NA | NA | PubChem |
| GABRA4 | Imidazoleacetic acid | NA | NA | NA | 340000 | NA | NA | BindingDB |
| GABRA4 | Tert-butyl 12-ethynyl-8-methyl-9-oxo-2,4,8-triazatricyclo[8.4.0.0^{2,6}]tetradeca-1(14),3,5,10,12-pentaene-5-carboxylate | NA | NA | NA | 324400 | NA | NA | BindingDB |
| GABRA5 | (4-Hydroxy-piperidin-4-yl)-phosphinic acid | 1900000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA5 | (Piperidin-4-yl)phosphonic acid | 2800000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA5 | (3-Aminopropyl)(n-butyl)phosphinic acid | NA | 508000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Delorazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Clonazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Nordazepam | NA | 106414000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Diazepam | NA | 123595000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Halazepam | NA | 10864300 | NA | NA | NA | NA | PubChem |
| GABRA5 | Flunitrazepam | NA | 263027000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Isonipecotic Acid | NA | NA | NA | 690000 | NA | NA | BindingDB |
| GABRA5 | Kynurenic Acid | NA | 2900000 | NA | NA | NA | NA | PubChem |
| GABRA5 | 3-Aminopropane-1-seleninic acid | NA | NA | NA | 1900000 | NA | NA | BindingDB |
| GABRA5 | Piperidine-4-Seleninic Acid | NA | NA | NA | 420000 | NA | NA | BindingDB |
| GABRA5 | Cocaine | NA | 127000 | NA | NA | NA | NA | PubChem |