Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| GABRA5 | Nitrazepam | NA | 100000000 | NA | NA | NA | NA | PubChem |
| GABRA5 | Temazepam | NA | 62517300 | NA | NA | NA | NA | PubChem |
| GABRA5 | Methyl(piperidin-4-yl)phosphinic acid | 420000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA5 | Piperidin-4-yl-phosphinic acid | NA | NA | NA | 260000 | NA | NA | BindingDB |
| GABRA5 | 7-Aminoflunitrazepam | NA | 15381500 | NA | NA | NA | NA | PubChem |
| GABRA5 | Imidazoleacetic acid | NA | NA | NA | 420000 | NA | NA | BindingDB |
| GABRA6 | (4-Hydroxy-piperidin-4-yl)-phosphinic acid | 3000000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA6 | (Piperidin-4-yl)phosphonic acid | 4800000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA6 | (3-Aminopropyl)(n-butyl)phosphinic acid | NA | 508000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Delorazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Clonazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Nordazepam | NA | 106414000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Diazepam | NA | 123595000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Halazepam | NA | 10864300 | NA | NA | NA | NA | PubChem |
| GABRA6 | Flunitrazepam | NA | 263027000 | NA | NA | NA | NA | PubChem |
| GABRA6 | Isonipecotic Acid | NA | NA | NA | 160000 | NA | NA | BindingDB |
| GABRA6 | Kynurenic Acid | NA | 2900000 | NA | NA | NA | NA | PubChem |
| GABRA6 | 3-Aminopropane-1-seleninic acid | NA | NA | NA | 3000000 | NA | NA | BindingDB |
| GABRA6 | Piperidine-4-Seleninic Acid | NA | NA | NA | 240000 | NA | NA | BindingDB |
| GABRA6 | Cocaine | NA | 127000 | NA | NA | NA | NA | PubChem |