Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| GABRQ | Delorazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRQ | Clonazepam | NA | 555904000 | NA | NA | NA | NA | PubChem |
| GABRQ | Nordazepam | NA | 106414000 | NA | NA | NA | NA | PubChem |
| GABRQ | Diazepam | NA | 123595000 | NA | NA | NA | NA | PubChem |
| GABRQ | Halazepam | NA | 10864300 | NA | NA | NA | NA | PubChem |
| GABRQ | Flunitrazepam | NA | 263027000 | NA | NA | NA | NA | PubChem |
| GABRQ | Cocaine | NA | 127000 | NA | NA | NA | NA | PubChem |
| GABRQ | Nitrazepam | NA | 100000000 | NA | NA | NA | NA | PubChem |
| GABRQ | Temazepam | NA | 62517300 | NA | NA | NA | NA | PubChem |
| GABRQ | 7-Aminoflunitrazepam | NA | 15381500 | NA | NA | NA | NA | PubChem |
| GABRR1 | 6-Amino-2-butylpyridine-3-carboxylic acid | NA | NA | NA | 1000000 | NA | NA | TTD |
| GABRR1 | 6-Amino-4-butylpyridine-3-carboxylic acid | NA | NA | NA | 1000000 | NA | NA | TTD |
| GABRR1 | (2R)-2-[(4S)-2-amino-4,5-dihydro-1,3-thiazol-4-yl]propanoic acid | NA | 300000 | NA | NA | NA | NA | BindingDB|TTD |
| GABRR1 | 6-Amino-2-ethylpyridine-3-carboxylic acid | NA | NA | NA | 1000000 | NA | NA | TTD |
| GABRR1 | 2-(2-amino-4-methyl-5H-1,3-thiazol-4-yl)acetic acid | NA | 300000 | NA | NA | NA | NA | BindingDB|TTD |
| GABRR1 | cis-2-Aminocyclopropanecarboxylic acid | NA | 890000 | NA | NA | NA | NA | BindingDB|TTD |
| GABRR1 | 6-Amino-4-ethylnicotinic acid | NA | NA | NA | 1000000 | NA | NA | TTD |
| GABRR1 | (5-Chloro-1-hydroxypyrazol-4-yl)methanamine | NA | NA | NA | 500000 | NA | NA | TTD |
| GABRR1 | (1-Hydroxy-3-iodopyrazol-4-yl)methanamine | NA | NA | NA | 500000 | NA | NA | TTD |
| GABRR1 | (3-Ethyl-1-hydroxypyrazol-4-yl)methanamine | NA | NA | NA | 500000 | NA | NA | TTD |