| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GABRR1 |
(1-Hydroxy-3-phenylpyrazol-4-yl)methanamine |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| GABRR1 |
[1-Hydroxy-3-(4-phenylphenyl)pyrazol-4-yl]methanamine |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| GABRR1 |
(1-Hydroxy-5-methylpyrazol-4-yl)methanamine |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| GABRR1 |
[1-Hydroxy-3-(3-phenylphenyl)pyrazol-4-yl]methanamine |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| GABRR1 |
4-amino-N-ethoxycyclopentene-1-carboxamide |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GABRR1 |
4-amino-N-prop-2-enoxycyclopentene-1-carboxamide |
NA |
115300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GABRR1 |
4-amino-N-methylcyclopentene-1-carboxamide |
NA |
408300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GABRR1 |
4-amino-N-propylcyclopentene-1-carboxamide |
NA |
570000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GABRR1 |
[(3S)-3-[6-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]hexanoylamino]cyclopenten-1-yl]-butylphosphinic acid |
NA |
147920 |
NA |
NA |
NA |
NA |
BindingDB |
| GABRR1 |
butyl-[(3S)-3-[6-[3-(2,2-difluoro-4,6,10,12-tetramethyl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-8-yl)propanoylamino]hexanoylamino]cyclopenten-1-yl]phosphinic acid |
NA |
103140 |
NA |
NA |
NA |
NA |
BindingDB |
| GABRR1 |
butyl-[(3S)-3-[6-[(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]hexanoylamino]cyclopenten-1-yl]phosphinic acid |
NA |
193270|281420 |
NA |
NA |
NA |
NA |
BindingDB |
| GABRR2 |
4-Amino-2-methylbut-2-enoic acid |
NA |
NA |
NA |
101000 |
NA |
NA |
BindingDB|TTD |
| GAK |
Sgcgak1N |
NA |
NA |
2500000 |
NA |
NA |
NA |
BindingDB |
| GALR2 |
2-[1-(3-bicyclo[2.2.1]heptanyl)tetrazol-5-yl]sulfanyl-N-quinolin-4-ylacetamide |
NA |
2529000 |
NA |
NA |
NA |
NA |
BindingDB |
| GALR2 |
4-Piperidin-1-yl-5H-pyrimido[5,4-b]indole |
NA |
108200 |
NA |
NA |
NA |
NA |
BindingDB |
| GALR2 |
4-butoxy-8-fluoro-5H-pyrimido[5,4-b]indole |
NA |
471500 |
NA |
NA |
NA |
NA |
BindingDB |
| GANAB |
(2R,3R,4R,5S)-2-Methylpiperidine-3,4,5-triol |
1560000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GANAB |
(2R,3R,4S)-2-ethylpyrrolidine-3,4-diol |
NA |
800000|1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| GANAB |
1-Deoxynojirimycin |
NA|410000|460000 |
210000|320000|500000|570000|NA|1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| GANAB |
(2R,3R,4R,5S)-2-(1-Hydroxy-propyl)-piperidine-3,4,5-triol |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |